SCHEMBL5162405

SCHEMBL5162405

CCC(Oc1ccccc1)C(=O)NC1CCC(Cc2ccccc2C)(N(C)C)CC1.CN(C)C1(Cc2cccc(F)c2)CCC(NC(=O)COc2ccc(Cl)cc2)CC1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PPARG P37231 2/20 0.39
PPARA Q07869 2/20 0.39
ATF4 P18848 3/20 0.39
MCHR1 Q99705 4/20 0.37
POLB P06746 1/20 0.36
USP2 O75604 1/20 0.36
LMNA P02545 1/20 0.35
SIGMAR1 Q99720 1/20 0.34
ADIPOR2 Q86V24 1/20 0.34
ADIPOR1 Q96A54 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2976658 0.84 MEN1 (0.45) PPARGPPARALMNASIGMAR1MEN1
SCHEMBL2972810 0.84 ATF4 (0.55) ATF4MCHR1POLBUSP2LMNA
SCHEMBL2989619 0.81 KMT2A (0.48) PPARGPPARAPOLBLMNAMEN1
SCHEMBL2989096 0.81 ATF4 (0.58) ATF4LMNAMEN1ALDH1A1KMT2A
SCHEMBL2987754 0.81 POLB (0.50) POLBUSP2LMNASIGMAR1ADIPOR2
SCHEMBL2982908 0.78 MCHR1 (0.50) ATF4MCHR1POLBLMNASIGMAR1
SCHEMBL2984841 0.78 LMNA (0.48) ATF4POLBLMNAMEN1ALDH1A1
SCHEMBL2987483 0.77 ATF4 (0.61) ATF4MCHR1POLBUSP2LMNA
SCHEMBL5162540 0.77 MCHR1 (0.46) MCHR1POLBSIGMAR1
SCHEMBL2981298 0.77 ATF4 (0.56) ATF4MCHR1POLBLMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1747191-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES WITH A CHAIN EXTENSION Grünenthal GmbH (DE) 2007-01-31 EP disclosed
WO-2005110975-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES WITH A CHAIN EXTENSION Grünenthal GmbH (DE) 2005-11-24 WO disclosed