SCHEMBL5162540

SCHEMBL5162540

CN(C)C1(CCc2ccccc2)CCC(NC(=O)COc2cccc(Cl)c2)CC1.CN(C)C1(Cc2cccc(F)c2)CCC(NC(=O)COc2ccccc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 15/20 0.46
POLB P06746 1/20 0.45
SIGMAR1 Q99720 1/20 0.42
KCNH2 Q12809 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2982908 0.93 MCHR1 (0.50) MCHR1POLBSIGMAR1KCNH2
SCHEMBL2976726 0.91 MCHR1 (0.54) MCHR1POLBSIGMAR1
SCHEMBL2987754 0.89 POLB (0.50) POLBSIGMAR1
SCHEMBL2983707 0.88 POLB (0.53) MCHR1POLBSIGMAR1
SCHEMBL2972810 0.87 ATF4 (0.55) MCHR1POLBSIGMAR1
SCHEMBL2987366 0.87 MCHR1 (0.54) MCHR1POLBKCNH2
SCHEMBL5162561 0.86 ALDH1A1 (0.40) POLBSIGMAR1
SCHEMBL2978691 0.83 MCHR1 (0.51) MCHR1POLB
SCHEMBL2972824 0.83 ATF4 (0.59) MCHR1POLB
SCHEMBL2987178 0.82 ATF4 (0.58) MCHR1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007536322-A 2007-12-13 JP claimed
EP-1747191-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES WITH A CHAIN EXTENSION Grünenthal GmbH (DE) 2007-01-31 EP claimed
WO-2005110975-A1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES WITH A CHAIN EXTENSION Grünenthal GmbH (DE) 2005-11-24 WO claimed