SCHEMBL5162450

SCHEMBL5162450

O=C(NC(c1c[nH]cn1)C1CCCCC1)OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.47
CYP1A2 P05177 4/20 0.46
EPHX1 P07099 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
CYP3A4 P08684 8/20 0.44
TSHR P16473 5/20 0.44
CYP2C9 P11712 4/20 0.43
CYP2C19 P33261 4/20 0.43
POLB P06746 1/20 0.43
CYP2D6 P10635 1/20 0.43
LMNA P02545 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
GAA P10253 1/20 0.42
CTSL P07711 1/20 0.42
CTSB P07858 1/20 0.42
CTSS P25774 1/20 0.42
CTSK P43235 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23038201 0.78 ATM (0.50) POLBCTSLCTSSCTSK
SCHEMBL22244421 0.75 ALDH1A1 (0.57) ALDH1A1CYP1A2EPHX1MEN1KMT2A
SCHEMBL2326093 0.74 ALDH1A1 (0.56) ALDH1A1CYP1A2EPHX1MEN1KMT2A
SCHEMBL22285596 0.74 ALDH1A1 (0.56) ALDH1A1CYP1A2EPHX1MEN1KMT2A
SCHEMBL433978 0.74 ALDH1A1 (0.56) ALDH1A1CYP1A2EPHX1MEN1KMT2A
SCHEMBL25447123 0.74 ALDH1A1 (0.56) ALDH1A1CYP1A2EPHX1MEN1KMT2A
SCHEMBL22285592 0.74 ALDH1A1 (0.56) ALDH1A1CYP1A2EPHX1MEN1KMT2A
SCHEMBL9398324 0.74 ALDH1A1 (0.56) ALDH1A1CYP1A2EPHX1MEN1KMT2A
SCHEMBL433979 0.74 ALDH1A1 (0.56) ALDH1A1CYP1A2EPHX1MEN1KMT2A
SCHEMBL5461377 0.74 ALDH1A1 (0.56) ALDH1A1CYP1A2CYP3A4TSHRCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765791-A1 PYRIMIDINE DERIVATIVES USEFUL AS INHIBITORS OF PKC-THETA BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2007-03-28 EP disclosed
WO-2006014482-A1 PYRIMIDINE DERIVATIVES USEFUL AS INHIBITORS OF PKC-THETA BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2006-02-09 WO disclosed