SCHEMBL5163030

SCHEMBL5163030

C=C(C)C(=O)NC(C)P(=O)(O)OCC

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 1/20 0.39
GAA P10253 1/20 0.34
MMP1 P03956 2/20 0.33
MMP2 P08253 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
MMP3 P08254 1/20 0.33
CA12 O43570 2/20 0.32
CA1 P00915 2/20 0.32
CA2 P00918 2/20 0.32
CA9 Q16790 2/20 0.32
PPARD Q03181 1/20 0.32
TSHR P16473 3/20 0.31
MMP8 P22894 1/20 0.31
ALDH1A1 P00352 2/20 0.31
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5165317 0.95 TGFBR1 (0.36) TGFBR1GAAMMP1MMP2CYP3A4
SCHEMBL976101 0.76 TGFBR1 (0.42) TGFBR1MMP1MMP2MMP3CA12
SCHEMBL976256 0.72 TGFBR1 (0.39) TGFBR1MMP1MMP2CYP2C19CA12
SCHEMBL28963627 0.71 LPAR3 (0.45) TGFBR1MMP1MMP2MMP3TSHR
SCHEMBL5697275 0.71 TSHR (0.39) PPARDTSHRALDH1A1
SCHEMBL184419 0.71 NPSR1 (0.37) TGFBR1GAACA12CA1CA2
SCHEMBL641337 0.69 TGFBR1 (0.44) TGFBR1GAATSHRALDH1A1
SCHEMBL4187674 0.69 FDPS (0.41) TGFBR1MMP1MMP2CA12CA1
SCHEMBL28963629 0.69 PPARD (0.33) TGFBR1GAACYP3A4CYP2C9CYP2C19
SCHEMBL14368417 0.69 TGFBR1 (0.41) TGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765895-A1 SYNTHESIS OF COPOLYMERS IN THE FORM OF A MIKTO STAR BY CONTROLLED RADICAL POLYMERIZATION RHODIA CHIMIE (FR) 2007-03-28 EP claimed
WO-2005116097-A1 SYNTHESIS OF COPOLYMERS IN THE FORM OF A MIKTO STAR BY CONTROLLED RADICAL POLYMERIZATION RHODIA CHIMIE (FR) 2005-12-08 WO claimed
EP-1527105-A2 SYNTHESIS OF STATISTICAL MICROGELS BY MEANS OF CONTROLLED RADICAL POLYMERISATION RHODIA CHIMIE (FR) 2005-05-04 EP claimed
EP-1483341-A1 USE OF BLOCK COPOLYMERS BEARING PHOSPHATE AND/OR PHOSPHONATE FUNCTIONS AS ADHESION PROMOTERS OR AS PROTECTING AGENTS AGAINST THE CORROSION OF A METALLIC SURFACE RHODIA CHIMIE (FR) 2004-12-08 EP claimed
EP-1483344-A1 USE OF BLOCK COPOLYMERS BEARING PHOSPHATE AND/OR PHOSPHONATE FUNCTIONS AS ADHESION PROMOTERS OR AS PROTECTING AGENTS AGAINST THE CORROSION OF A METALLIC SURFACE RHODIA CHIMIE (FR) 2004-12-08 EP claimed
WO-2004014535-A2 SYNTHESIS OF STATISTICAL MICROGELS BY MEANS OF CONTROLLED RADICAL POLYMERISATION RHODIA CHIMIE (FR) 2004-02-19 WO claimed
WO-2003076531-A1 USE OF BLOCK COPOLYMERS BEARING PHOSPHATE AND/OR PHOSPHONATE FUNCTIONS AS ADHESION PROMOTERS OR AS PROTECTING AGENTS AGAINST THE CORROSION OF A METALLIC SURFACE RHODIA CHIMIE (FR) 2003-09-18 WO claimed
WO-2003076529-A1 USE OF BLOCK COPOLYMERS BEARING PHOSPHATE AND/OR PHOSPHONATE FUNCTIONS AS ADHESION PROMOTERS OR AS PROTECTING AGENTS AGAINST THE CORROSION OF A METALLIC SURFACE RHODIA CHIMIE (FR) 2003-09-18 WO claimed
WO-2023110696-A1 METHOD FOR THE EMULSION POLYMERIZATION OF FLUOROMONOMER SOLVAY SPECIALTY POLYMERS ITALY S.P.A. (IT) 2023-06-22 WO disclosed
EP-2838816-A1 LOW VOC, WATER-BASED COATING COMPOSITIONS SUITABLE FOR PROTECTING METAL CONTAINING SUBSTRATES INCLUDING FOOD AND BEVERAGE PACKAGES Valspar Sourcing, Inc. (US) 2015-02-25 EP disclosed
WO-2013158261-A1 LOW VOC, WATER-BASED COATING COMPOSITIONS SUITABLE FOR PROTECTING METAL CONTAINING SUBSTRATES INCLUDING FOOD AND BEVERAGE PACKAGES VALSPAR CORPORATION (US) 2013-10-24 WO disclosed
EP-1527105-A2 SYNTHESIS OF STATISTICAL MICROGELS BY MEANS OF CONTROLLED RADICAL POLYMERISATION RHODIA CHIMIE (FR) 2005-05-04 EP disclosed
EP-1483341-A1 USE OF BLOCK COPOLYMERS BEARING PHOSPHATE AND/OR PHOSPHONATE FUNCTIONS AS ADHESION PROMOTERS OR AS PROTECTING AGENTS AGAINST THE CORROSION OF A METALLIC SURFACE RHODIA CHIMIE (FR) 2004-12-08 EP disclosed
EP-1483344-A1 USE OF BLOCK COPOLYMERS BEARING PHOSPHATE AND/OR PHOSPHONATE FUNCTIONS AS ADHESION PROMOTERS OR AS PROTECTING AGENTS AGAINST THE CORROSION OF A METALLIC SURFACE RHODIA CHIMIE (FR) 2004-12-08 EP disclosed
WO-2004014535-A2 SYNTHESIS OF STATISTICAL MICROGELS BY MEANS OF CONTROLLED RADICAL POLYMERISATION RHODIA CHIMIE (FR) 2004-02-19 WO disclosed
WO-2003076531-A1 USE OF BLOCK COPOLYMERS BEARING PHOSPHATE AND/OR PHOSPHONATE FUNCTIONS AS ADHESION PROMOTERS OR AS PROTECTING AGENTS AGAINST THE CORROSION OF A METALLIC SURFACE RHODIA CHIMIE (FR) 2003-09-18 WO disclosed
WO-2003076529-A1 USE OF BLOCK COPOLYMERS BEARING PHOSPHATE AND/OR PHOSPHONATE FUNCTIONS AS ADHESION PROMOTERS OR AS PROTECTING AGENTS AGAINST THE CORROSION OF A METALLIC SURFACE RHODIA CHIMIE (FR) 2003-09-18 WO disclosed