SCHEMBL5164396

SCHEMBL5164396

Cc1ccc(C(CO)[N+](=O)[O-])cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.42
HSD17B10 Q99714 1/20 0.42
GAA P10253 3/20 0.40
ALDH1A1 P00352 4/20 0.39
MAPT P10636 3/20 0.39
HSP90AA1 P07900 2/20 0.39
MAPK1 P28482 1/20 0.39
AGTR1 P30556 1/20 0.39
ATM Q13315 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
HPGD P15428 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
FBP1 P09467 1/20 0.36
LMNA P02545 1/20 0.36
GSR P00390 1/20 0.36
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
CYP3A4 P08684 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11040665 0.92 GAA (0.39) ACHEHSD17B10GAAALDH1A1MAPT
SCHEMBL9337987 0.82 ACHE (0.43) ACHEHSD17B10GAAALDH1A1MAPT
SCHEMBL2461330 0.81 IGF1R (0.37) ALDH1A1MAPTATMLMNAGSR
SCHEMBL6258107 0.81 ALDH1A1 (0.53) ACHEHSD17B10ALDH1A1MAPTMAPK1
SCHEMBL2461283 0.81 IGF1R (0.37) ALDH1A1MAPTATMLMNAGSR
SCHEMBL28306985 0.81 ALDH1A1 (0.42) HSD17B10ALDH1A1MAPTHSP90AA1MAPK1
SCHEMBL3336779 0.80 GSR (0.55) ALDH1A1MAPTMAPK1NPSR1TDP1
Fluoride SCHEMBL28046654 0.78 GSR (0.53) ALDH1A1MAPTMAPK1NPSR1TDP1
SCHEMBL4269735 0.78 MAPT (0.41) ACHEHSD17B10GAAALDH1A1MAPT
SCHEMBL11043092 0.75 GSR (0.46) ALDH1A1MAPTMAPK1NPSR1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765793-A1 CETP INHIBITORS Merck and Co., Inc. (US) 2007-03-28 EP disclosed
WO-2006014357-A1 CETP INHIBITORS MERCK & CO., INC. (US) 2006-02-09 WO disclosed
WO-2006014413-A1 CETP INHIBITORS MERCK & CO., INC. (US) 2006-02-09 WO disclosed