SCHEMBL5165075

SCHEMBL5165075

CC(C)=CCc1cc(CC=O)c(O)c(CC=C(C)C)c1O

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.66
KMT2A Q03164 2/20 0.66
TRPV4 Q9HBA0 1/20 0.49
AKR1B10 O60218 1/20 0.47
MMP2 P08253 1/20 0.47
AKR1B1 P15121 1/20 0.47
AKR1C3 P42330 1/20 0.47
PAK1 Q13153 1/20 0.47
MAOB P27338 1/20 0.47
HTT P42858 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
HPGD P15428 1/20 0.44
CYP2C19 P33261 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
CNR1 P21554 1/20 0.43
CNR2 P34972 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29249591 0.82 MEN1 (0.42) MEN1KMT2ATRPV4AKR1B10MMP2
SCHEMBL5166422 0.82 AKR1B10 (0.51) MEN1KMT2ATRPV4AKR1B10MMP2
SCHEMBL5165720 0.81 AKR1B10 (0.54) MEN1KMT2ATRPV4AKR1B10MMP2
Methane SCHEMBL27993257 0.81 MEN1 (0.60) MEN1KMT2ATRPV4AKR1B10MMP2
SCHEMBL4104687 0.79 MEN1 (1.00) MEN1KMT2ATRPV4AKR1B10MMP2
SCHEMBL27028792 0.76 CYP19A1 (0.51) MEN1KMT2AAKR1B1MAOBHTT
SCHEMBL11116300 0.75 MEN1 (0.40) MEN1KMT2ATRPV4MAOBHTT
SCHEMBL30199523 0.74 AKR1B10 (0.63) MEN1KMT2AAKR1B10MMP2AKR1B1
SCHEMBL12733155 0.72 AKR1B10 (0.56) MEN1KMT2ATRPV4AKR1B10MMP2
SCHEMBL7898977 0.72 CYP19A1 (0.55) MEN1KMT2AAKR1B1MAOBHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1768945-A1 SUBSTITUTED HYDROXYACETOPHENON DERIVATIVES Riemser Arzneimittel AG (DE) 2007-04-04 EP claimed
WO-2006003010-A1 SUBSTITUTED HYDROXYACETOPHENON DERIVATIVES RIEMSER ARZNEIMITTEL AG (DE) 2006-01-12 WO claimed
EP-1768945-A1 SUBSTITUTED HYDROXYACETOPHENON DERIVATIVES Riemser Arzneimittel AG (DE) 2007-04-04 EP disclosed
WO-2006003010-A1 SUBSTITUTED HYDROXYACETOPHENON DERIVATIVES RIEMSER ARZNEIMITTEL AG (DE) 2006-01-12 WO disclosed