SCHEMBL5165286

SCHEMBL5165286

COc1c(F)c(F)cc2c(=O)c(OC(=O)OCC(F)(F)F)c[nH]c12

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.33
LMNA P02545 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C19 P33261 1/20 0.32
ALDH1A1 P00352 2/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5029833 0.78 LRRK2 (0.32) KDM4EALDH1A1HPGD
SCHEMBL5029782 0.78 KCNH2 (0.32) KDM4EALDH1A1HPGD
SCHEMBL1345017 0.74 CYP1A2 (0.59) KDM4ECYP1A2CYP3A4CYP2C19ALDH1A1
SCHEMBL20258340 0.73 CYP1A2 (0.42) KDM4ELMNACYP1A2CYP3A4CYP2C19
SCHEMBL8559994 0.72 CYP1A2 (0.40) KDM4ELMNACYP1A2CYP3A4CYP2C19
SCHEMBL9535556 0.71 ALDH1A1 (0.48) KDM4ELMNACYP1A2ALDH1A1HPGD
SCHEMBL8561725 0.70 CYP1A2 (0.38) KDM4ELMNACYP1A2CYP3A4CYP2C19
SCHEMBL6584701 0.68 HTR3E (0.43) KDM4ELMNACYP1A2CYP3A4CYP2C19
SCHEMBL1973321 0.68 STAT3 (0.40) KDM4EALDH1A1HPGD
SCHEMBL4735055 0.67 ALDH1A1 (0.48) ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1768973-A1 SUBSTITUTED QUINOLONES AiCuris GmbH & Co. KG (DE) 2007-04-04 EP disclosed
WO-2006008046-A1 SUBSTITUTED QUINOLONES AICURIS GMBH & CO. KG (DE) 2006-01-26 WO disclosed