SCHEMBL8559994

SCHEMBL8559994

CCCc1c(F)c(F)cc2c(=O)c(OC(=O)OCC)c[nH]c12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C19 P33261 1/20 0.40
CLEC4M Q9H2X3 1/20 0.38
KDM4E B2RXH2 4/20 0.36
TYMS P04818 1/20 0.35
KMT2A Q03164 4/20 0.35
MEN1 O00255 3/20 0.35
CRHBP P24387 1/20 0.35
CRHR2 Q13324 1/20 0.35
LMNA P02545 2/20 0.34
MAPT P10636 2/20 0.34
CUL4A Q13619 2/20 0.33
ALDH1A1 P00352 2/20 0.33
TP53 P04637 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
STAT3 P40763 1/20 0.33
GABRA1 P14867 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8561725 0.81 CYP1A2 (0.38) CYP1A2CYP3A4CYP2C19CLEC4MKDM4E
SCHEMBL10766497 0.76 CYP1A2 (0.57) CYP1A2CYP3A4CYP2C19CLEC4MKDM4E
SCHEMBL8558746 0.75 KDM4E (0.46) CYP1A2CYP3A4CYP2C19KDM4EKMT2A
SCHEMBL8556453 0.74 CYP1A2 (0.36) CYP1A2CYP3A4CYP2C19CLEC4MKDM4E
SCHEMBL5165286 0.72 KDM4E (0.33) CYP1A2CYP3A4CYP2C19KDM4ELMNA
SCHEMBL9635290 0.71 CYP1A2 (0.66) CYP1A2CYP3A4CYP2C19CLEC4MKDM4E
SCHEMBL29376920 0.71 CYP1A2 (0.66) CYP1A2CYP3A4CYP2C19CLEC4MKDM4E
SCHEMBL8556198 0.70 MEN1 (0.39) KDM4EKMT2AMEN1LMNAMAPT
SCHEMBL7218429 0.70 NQO2 (0.40) CYP1A2CYP2C19KMT2AMEN1LMNA
SCHEMBL8318286 0.70 LMNA (0.35) CYP1A2CYP3A4CYP2C19KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0828715-A1 N-OXIDES AS ANTIBACTERIAL AGENTS BAYER AG (DE) 1998-03-18 EP disclosed
WO-1996038417-A1 N-OXIDES AS ANTIBACTERIAL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1996-12-05 WO disclosed