SCHEMBL5165517

SCHEMBL5165517

CCC(=O)CCCCC[C@H](NC(=O)C[S+](C)[O-])C(=O)NC1CCN(Cc2ccccc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR8 P51685 1/20 0.46
SIGMAR1 Q99720 9/20 0.45
CYP2C19 P33261 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
USP2 O75604 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5124876 0.89 SIGMAR1 (0.57) CCR8SIGMAR1
SCHEMBL5130455 0.87 BCHE (0.49) CCR8SIGMAR1CYP2C19SMN1; SMN2USP2
SCHEMBL5117306 0.86 CCR8 (0.47) CCR8SIGMAR1CYP2C19SMN1; SMN2USP2
SCHEMBL5118332 0.86 CCR8 (0.47) CCR8SIGMAR1CYP2C19SMN1; SMN2USP2
SCHEMBL5126563 0.84 CCR2 (0.53) SMN1; SMN2
SCHEMBL5121666 0.82 CYP2C19 (0.53) SIGMAR1CYP2C19SMN1; SMN2CYP2D6CYP2C9
SCHEMBL5164015 0.82 HDAC1 (0.48) SMN1; SMN2
SCHEMBL5119081 0.82 CCR8 (0.45) CCR8SIGMAR1CYP2C19SMN1; SMN2USP2
SCHEMBL5127760 0.80 SIGMAR1 (0.51) SIGMAR1SMN1; SMN2
SCHEMBL12488466 0.79 ALDH1A1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1768955-A1 AMIDE DERIVATIVES AS INHIBITORS OF HISTONE DEACETYLASE ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.P.A. (IT) 2007-04-04 EP disclosed
WO-2006005941-A1 AMIDE DERIVATIVES AS INHIBITORS OF HISTONE DEACETYLASE ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P ANGELETTI S.P.A. (IT) 2006-01-19 WO disclosed