SCHEMBL5165904

SCHEMBL5165904

CSc1cc(N)ccc1N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 5/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 1/20 0.43
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
ALDH1A1 P00352 4/20 0.40
KEAP1 Q14145 1/20 0.38
G6PD P11413 1/20 0.38
IDE P14735 1/20 0.38
CYP3A4 P08684 6/20 0.37
MEN1 O00255 5/20 0.37
KMT2A Q03164 5/20 0.37
MAPT P10636 4/20 0.37
POLB P06746 3/20 0.37
TDP1 Q9NUW8 3/20 0.37
RECQL P46063 3/20 0.37
ALOX15 P16050 3/20 0.37
THRB P10828 3/20 0.37
USP2 O75604 2/20 0.37
PKM P14618 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8448289 0.97 CASP1 (0.42) CASP1NPC1RAB9APTGS1PTGS2
Hydrochloric Acid SCHEMBL8448284 0.97 CASP1 (0.42) CASP1NPC1RAB9APTGS1PTGS2
SCHEMBL3783187 0.84 AAK1 (0.48) NPC1RAB9AALDH1A1CYP3A4MEN1
SCHEMBL11528651 0.82 AAK1 (0.50) NPC1RAB9AALDH1A1G6PDIDE
SCHEMBL8920417 0.82 CASP1 (0.48) CASP1NPC1RAB9APTGS1PTGS2
SCHEMBL9781542 0.82 NPC1 (0.63) NPC1RAB9AALDH1A1CYP3A4MEN1
SCHEMBL17498342 0.81 ITGB2 (0.43) CASP1NPC1RAB9AALDH1A1G6PD
SCHEMBL30678438 0.80 ALDH1A1 (0.54) CASP1NPC1RAB9APTGS1PTGS2
SCHEMBL9180206 0.80 NPC1 (0.41) NPC1RAB9AALDH1A1G6PDIDE
SCHEMBL8491702 0.80 ALDH1A1 (0.54) CASP1NPC1RAB9APTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1335900-B1 ALKYLTHIO- AND ARYL(HETEROYL)THIO-SUBSTITUTED P-PHENYLENEDIAMINES, THEIR MANUFACTURE AND THEIR USE IN RUBBER FLEXSYS AMERICA LP (US) 2007-04-18 EP claimed
EP-0656202-B1 Dyeing composition containing sulphurous p-phenylene-diamines, sulphurous p-phenylenediamines and method of preparation OREAL (FR) 1999-05-06 EP claimed
US-5542952-A DEVELOPERS THAT FORM STABLE OXIDATION HAIR DYES L'OREAL (FR) 1996-08-06 US claimed
EP-0656202-A1 Dyeing composition containing sulphurous p-phenylene-diamines, novel sulphurous p-phenylenediamines and method of preparation L'OREAL (FR) 1995-06-07 EP claimed
CN-114502672-A Coating composition PRC-迪索托国际公司 2022-05-13 CN disclosed
WO-2020059048-A1 SET COMPRISING MAIN AGENT AND CURING AGENT, WATER-RESISTANT MATERIAL, AND METHOD OF CONSTRUCTING SAME 保土谷化学工業株式会社 2020-03-26 WO disclosed
EP-1335900-B1 ALKYLTHIO- AND ARYL(HETEROYL)THIO-SUBSTITUTED P-PHENYLENEDIAMINES, THEIR MANUFACTURE AND THEIR USE IN RUBBER FLEXSYS AMERICA LP (US) 2007-04-18 EP disclosed
EP-0656202-B1 Dyeing composition containing sulphurous p-phenylene-diamines, sulphurous p-phenylenediamines and method of preparation OREAL (FR) 1999-05-06 EP disclosed
US-5542952-A DEVELOPERS THAT FORM STABLE OXIDATION HAIR DYES L'OREAL (FR) 1996-08-06 US disclosed
EP-0656202-A1 Dyeing composition containing sulphurous p-phenylene-diamines, novel sulphurous p-phenylenediamines and method of preparation L'OREAL (FR) 1995-06-07 EP disclosed
US-4239708-A P-Phenylene bis[imino(thiocarbonyl)] diphosphoramidic acid esters as anthelmentic agents AMERICAN CYANAMID COMPANY (US) 1980-12-16 US disclosed
EP-0001604-B1 AROMATIC DIISOCYANATES, PROCESS FOR THEIR PREPARATION AND THEIR USE IN THE PREPARATION OF POLYURETHANES BAYER AG (DE) 1980-07-23 EP disclosed
EP-0001604-A2 Aromatic diisocyanates, process for their preparation and their use in the preparation of polyurethanes BAYER AG (DE) 1979-05-02 EP disclosed
US-4137310-A LARVICIDES AMERICAN CYANAMID COMPANY (US) 1979-01-30 US disclosed