SCHEMBL5165973

SCHEMBL5165973

C[Si](C)(C)C#Cc1ccc(OCc2cccnc2)c(N)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.42
HTR1A P08908 2/20 0.41
DRD2 P14416 2/20 0.41
NOS3 P29474 1/20 0.41
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41
MRGPRX1 Q96LB2 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CYP11B1 P15538 2/20 0.40
CYP11B2 P19099 2/20 0.40
CYP19A1 P11511 1/20 0.40
CHEK1 O14757 1/20 0.40
IKBKB O14920 1/20 0.40
SLC6A4 P31645 1/20 0.39
ACACB O00763 2/20 0.39
PRKDC P78527 1/20 0.39
PTAFR P25105 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
P2RY12 Q9H244 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5165371 0.81 LMNA (0.44) LMNACYP11B1CYP11B2CYP19A1ACACB
SCHEMBL2038082 0.78 LRRK2 (0.50) LMNAHTR1ADRD2NOS3NOS1
SCHEMBL13428030 0.78 CYP19A1 (0.58) LMNAHTR1ADRD2NOS3NOS1
SCHEMBL17323482 0.76 HTR1A (0.54) LMNAHTR1ADRD2NOS3NOS1
SCHEMBL2038362 0.76 HTR1A (0.51) HTR1ADRD2NOS3NOS1NOS2
SCHEMBL1028598 0.73 HTR1A (0.61) HTR1ADRD2NOS3NOS1NOS2
SCHEMBL30697112 0.73 HTR1A (0.43) LMNAHTR1ADRD2HSD17B10CYP11B1
SCHEMBL22711531 0.73 HTR1A (0.43) LMNAHTR1ADRD2HSD17B10CYP11B1
SCHEMBL5164933 0.73 CHEK1 (0.49) HSD17B10CHEK1ACACB
SCHEMBL17629916 0.73 CYP11B1 (0.50) HTR1ADRD2NOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765808-A1 BISARYLUREA DERIVATIVES USEFUL FOR INHIBITING CHK1 ICOS Corporation (US) 2007-03-28 EP disclosed
WO-2006012308-A1 BISARYLUREA DERIVATIVES USEFUL FOR INHIBITING CHK1 ICOS CORPORATION (US) 2006-02-02 WO disclosed