SCHEMBL5166106

SCHEMBL5166106

O=C(O)C1CCC(CCN(Cc2ccccc2)Cc2ccccc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
TAS2R14 Q9NYV8 7/20 0.49
L3MBTL1 Q9Y468 1/20 0.43
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
HDAC3 O15379 2/20 0.42
HDAC1 Q13547 2/20 0.42
HDAC2 Q92769 2/20 0.42
HDAC8 Q9BY41 2/20 0.42
NCOR2 Q9Y618 2/20 0.42
ACHE P22303 2/20 0.42
KDM4E B2RXH2 1/20 0.42
HSD17B10 Q99714 1/20 0.42
POLB P06746 1/20 0.41
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22482261 0.87 KDM4E (0.46) MEN1KMT2AL3MBTL1ALDH1A1HDAC3
SCHEMBL4479586 0.84 TAS2R14 (0.57) MEN1KMT2ATAS2R14L3MBTL1ALDH1A1
SCHEMBL4479581 0.84 TAS2R14 (0.57) MEN1KMT2ATAS2R14L3MBTL1ALDH1A1
SCHEMBL785821 0.79 ACHE (0.49) ACHE
SCHEMBL7814243 0.79 POLB (0.54) TAS2R14L3MBTL1ALDH1A1GAAKDM4E
SCHEMBL1965678 0.79 TAS2R14 (0.49) MEN1KMT2ATAS2R14L3MBTL1ALDH1A1
SCHEMBL784983 0.76 GBA1 (0.56) KDM4EHSD17B10
Trifluoroacetic Acid SCHEMBL785809 0.76 SLC6A2 (0.46) MEN1KMT2A
SCHEMBL3515654 0.75 GBA1 (0.53) MEN1KMT2AL3MBTL1ALDH1A1GAA
SCHEMBL1662783 0.75 GBA1 (0.53) MEN1KMT2AL3MBTL1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765791-A1 PYRIMIDINE DERIVATIVES USEFUL AS INHIBITORS OF PKC-THETA BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2007-03-28 EP disclosed
WO-2006014482-A1 PYRIMIDINE DERIVATIVES USEFUL AS INHIBITORS OF PKC-THETA BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2006-02-09 WO disclosed