SCHEMBL5166162

SCHEMBL5166162

C=C(CN(C)Cc1ccc(C(C)(C)C)cc1)c1ccccc1[N+](=O)[O-]

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.47
MAPT P10636 2/20 0.46
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
LMNA P02545 3/20 0.40
SIGMAR1 Q99720 2/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
NR1I2 O75469 1/20 0.40
ADRA2A P08913 1/20 0.40
CYP2D6 P10635 1/20 0.40
ACHE P22303 1/20 0.40
SLC6A2 P23975 1/20 0.40
HTR2A P28223 1/20 0.40
SLC6A4 P31645 1/20 0.40
KCNH2 Q12809 1/20 0.40
TP53 P04637 1/20 0.40
PTPN1 P18031 1/20 0.39
TMEM97 Q5BJF2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5168222 0.87 NPSR1 (0.50) NPSR1MAPTALDH1A1KDM4EL3MBTL1
SCHEMBL5165584 0.80 SIGMAR1 (0.45) LMNASIGMAR1KMT2AMEN1NR1I2
SCHEMBL5167008 0.79 SIGMAR1 (0.44) ALDH1A1KDM4EL3MBTL1LMNASIGMAR1
SCHEMBL5167060 0.79 SIGMAR1 (0.44) KDM4ELMNASIGMAR1KMT2AMEN1
SCHEMBL5169554 0.79 MAPT (0.48) NPSR1MAPTALDH1A1LMNASIGMAR1
SCHEMBL5166525 0.77 ALDH1A1 (0.46) MAPTALDH1A1L3MBTL1LMNASIGMAR1
SCHEMBL5169309 0.77 MAPT (0.46) NPSR1MAPTKDM4ELMNASIGMAR1
SCHEMBL5165543 0.76 MAOA (0.50) MAPTL3MBTL1LMNASIGMAR1KMT2A
Hydrochloric Acid SCHEMBL5168719 0.75 MAOA (0.51) LMNASIGMAR1KMT2AMEN1NR1I2
SCHEMBL5166710 0.74 SIGMAR1 (0.45) LMNASIGMAR1NR1I2ADRA2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1561744-B1 AMINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND THEIR USE AS ANTIMYCOTIC AGENT POLA CHEM IND INC (JP) 2007-04-18 EP claimed
EP-1561744-A2 AMINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND THEIR USE AS ANTIMYCOTIC AGENT POLA CHEMICAL INDUSTRIES INC. (JP) 2005-08-10 EP claimed
US-6329399-B1 Antifungal amine derivatives and processing for producing the same POLA CHEMICAL INDUSTRIES, INC. (JP) 2001-12-11 US claimed
EP-1020426-A1 AMINE DERIVATIVES AND PROCESS FOR PRODUCING THE SAME POLA CHEMICAL INDUSTRIES, INC. (JP) 2000-07-19 EP claimed
EP-1561744-B1 AMINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND THEIR USE AS ANTIMYCOTIC AGENT POLA CHEM IND INC (JP) 2007-04-18 EP disclosed
EP-1561744-A2 AMINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND THEIR USE AS ANTIMYCOTIC AGENT POLA CHEMICAL INDUSTRIES INC. (JP) 2005-08-10 EP disclosed
US-6329399-B1 Antifungal amine derivatives and processing for producing the same POLA CHEMICAL INDUSTRIES, INC. (JP) 2001-12-11 US disclosed
EP-1020426-A1 AMINE DERIVATIVES AND PROCESS FOR PRODUCING THE SAME POLA CHEMICAL INDUSTRIES, INC. (JP) 2000-07-19 EP disclosed