SCHEMBL5167311

SCHEMBL5167311

COc1ccccc1S(=O)(=O)N(Cc1ccc(-c2ccc3c(c2)COC3)cc1)Cc1ccc(CP(=O)(OF)OF)c(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 6/20 0.39
NR1H3 Q13133 5/20 0.39
ACLY P53396 1/20 0.34
EP300 Q09472 1/20 0.33
HIF1A Q16665 1/20 0.33
HTT P42858 2/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
ALDH1A1 P00352 5/20 0.32
TAS2R14 Q9NYV8 3/20 0.32
KCNA5 P22460 1/20 0.32
BDKRB1 P46663 1/20 0.31
KDM4E B2RXH2 2/20 0.31
HSD17B10 Q99714 2/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
HPGD P15428 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5178441 0.89 NR1H2 (0.38) NR1H2NR1H3ACLYEP300HIF1A
SCHEMBL5166577 0.84 ALDH1A1 (0.41) NR1H2NR1H3ACLYHTTLMNA
SCHEMBL5163077 0.83 LMNA (0.40) NR1H2NR1H3ACLYHTTLMNA
SCHEMBL5167005 0.83 NR1H2 (0.42) NR1H2NR1H3ACLYHIF1ALMNA
SCHEMBL5164531 0.82 NR1H2 (0.40) NR1H2NR1H3ACLYHTTLMNA
SCHEMBL5165874 0.82 ACLY (0.44) NR1H2NR1H3ACLYHTTLMNA
SCHEMBL5164817 0.82 PTPN1 (0.42) NR1H2NR1H3ACLYHTTLMNA
SCHEMBL5164630 0.82 ACLY (0.42) NR1H2NR1H3ACLYHTTLMNA
SCHEMBL5165472 0.81 GSK3B (0.37) NR1H2NR1H3MAPTNPSR1ALDH1A1
SCHEMBL5163888 0.81 ALDH1A1 (0.42) LMNANPSR1ALDH1A1TAS2R14KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765332-A2 TRISUBSTITUTED NITROGEN MODULATORS OF TYROSINE PHOSPHATASES Cengent Therapeutics, Inc. (US) 2007-03-28 EP disclosed
WO-2006009876-A2 TRISUBSTITUTED NITROGEN MODULATORS OF TYROSINE PHOSPHATASES CENGENT THERAPEUTICS, INC. (US) 2006-01-26 WO disclosed