SCHEMBL5167844

SCHEMBL5167844

O=[N+]([O-])c1cccc2cc3cc4ccccc4cc3cc12

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.66
TDP1 Q9NUW8 3/20 0.57
CYP3A4 P08684 1/20 0.55
TSHR P16473 1/20 0.53
CASP6 P55212 1/20 0.51
HPRT1 P00492 1/20 0.47
GPR35 Q9HC97 1/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
RAB9A P51151 1/20 0.45
MAOA P21397 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
PDE10A Q9Y233 1/20 0.44
HSD17B10 Q99714 1/20 0.44
NOS1 P29475 1/20 0.44
NOS2 P35228 1/20 0.44
POLB P06746 1/20 0.43
CTSB P07858 1/20 0.43
CDK2 P24941 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL579426 0.98 ALDH1A1 (0.68) ALDH1A1TDP1CYP3A4TSHRCASP6
SCHEMBL30696914 0.98 ALDH1A1 (0.68) ALDH1A1TDP1CYP3A4TSHRCASP6
SCHEMBL9735773 0.92 ALDH1A1 (0.69) ALDH1A1TDP1CYP3A4TSHRCASP6
SCHEMBL9734521 0.90 ALDH1A1 (0.67) ALDH1A1TDP1CYP3A4TSHRCASP6
Benzoquinone SCHEMBL28192198 0.90 ALDH1A1 (0.58) ALDH1A1TDP1CYP3A4TSHRCASP6
SCHEMBL28197400 0.88 TDP1 (0.54) ALDH1A1TDP1CYP3A4TSHRCASP6
SCHEMBL28257118 0.88 TDP1 (0.54) ALDH1A1TDP1CYP3A4TSHRCASP6
Naphthoquinone SCHEMBL28243040 0.85 ALDH1A1 (0.53) ALDH1A1TDP1CYP3A4TSHRCASP6
SCHEMBL14183908 0.84 ALDH1A1 (0.55) ALDH1A1TDP1CYP3A4TSHRCASP6
SCHEMBL28749541 0.84 ALDH1A1 (0.55) ALDH1A1TDP1CYP3A4TSHRCASP6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7250438-B2 Anti-bacterial and anti-cancer spiro beta-lactone/gamma-lactams NEREUS PHARMACEUTICALS, INC. (US) 2007-07-31 US disclosed
WO-2005121148-A9 ANTI-BACTERIAL AND ANTI-CANCER SPIRO BETA-LACTONE/GAMMA-LACTAMS 2006-04-27 WO disclosed
US-20060004079-A1 Anti-bacterial and anti-cancer spiro beta-lactone/gamma-lactams PACIFIC VENTURE GROUP II, L.P. 2006-01-05 US disclosed
WO-2005121148-A2 ANTI-BACTERIAL AND ANTI-CANCER SPIRO BETA-LACTONE/GAMMA-LACTAMS NEREUS PHARMACEUTICALS, INC. (US) 2005-12-22 WO disclosed
EP-0649022-B1 Optical indicator for determining the activity of an ion in a sample AVL MEDICAL INSTR AG (CH) 1998-11-04 EP disclosed
EP-0705244-B1 NITRATO AMINO ACID DISULPHIDES FOR USE IN THE THERAPY OF DISORDERS OF THE CARDIOVASCULARY SYSTEM SANOL ARZNEI SCHWARZ GMBH (DE) 1998-11-04 EP disclosed
US-5723340-A COMPLEXING DIAMIDE IONOPHORE WITH LITHIUM, SODIUM, MAGNESIUM, OR CALCIUM; FLUORESCENCE AVL MEDICAL INSTRUMENTS AG (CH) 1998-03-03 US disclosed
EP-0705244-A1 NITRATO AMINO ACID DISULPHIDES FOR USE IN THE THERAPY OF DISORDERS OF THE CARDIOVASCULARY SYSTEM SCHWARZ PHARMA AG (DE) 1996-04-10 EP disclosed
EP-0649022-A1 Optical indicator for determining the activity of an ion in a sample AVL Medical Instruments AG (CH) 1995-04-19 EP disclosed
WO-1995000477-A1 NITRATO AMINO ACID DISULPHIDES FOR USE IN THE THERAPY OF DISORDERS OF THE CARDIOVASCULARY SYSTEM SCHWARZ PHARMA AG (DE) 1995-01-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060004079-A1 Anti-bacterial and anti-cancer spiro beta-lactone/gamma-lactams GLB1, PGLS, LBR ALDH1A1 1675/4885TDP1 4133/4885CYP3A4 3135/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.