SCHEMBL5168748

SCHEMBL5168748

C=C(CN(C)Cc1cccc2ccccc12)c1ccc(C(C)(C)C)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.64
LMNA P02545 3/20 0.64
SLC6A2 P23975 3/20 0.64
SIGMAR1 Q99720 3/20 0.64
ADRA2A P08913 2/20 0.64
NR1I2 O75469 2/20 0.64
HTR2A P28223 2/20 0.64
SLC6A4 P31645 2/20 0.64
KCNH2 Q12809 2/20 0.64
ACHE P22303 1/20 0.64
CYP1A2 P05177 2/20 0.54
CYP2C19 P33261 2/20 0.54
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
HPGD P15428 1/20 0.49
CYP19A1 P11511 1/20 0.44
SQLE Q14534 1/20 0.44
HIF1A Q16665 2/20 0.42
DRD2 P14416 1/20 0.42
ADRA2C P18825 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5168255 0.87 CYP2D6 (0.63) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
SCHEMBL5167194 0.85 CYP2D6 (0.64) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
Butenafine SCHEMBL20456391 0.79 CYP2D6 (1.00) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
Butenafine SCHEMBL29354083 0.79 CYP2D6 (1.00) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
Butenafine SCHEMBL65526 0.79 CYP2D6 (1.00) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
Butenafine SCHEMBL29459249 0.78 LMNA (0.97) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
Butenafine SCHEMBL676912 0.78 LMNA (0.97) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
Butenafine SCHEMBL262301 0.78 LMNA (0.97) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
SCHEMBL5169170 0.78 PYCR1 (0.46) CYP2D6LMNASLC6A2SIGMAR1ADRA2A
SCHEMBL1931930 0.77 CYP2D6 (0.69) CYP2D6LMNASLC6A2SIGMAR1ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1561744-B1 AMINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND THEIR USE AS ANTIMYCOTIC AGENT POLA CHEM IND INC (JP) 2007-04-18 EP claimed
US-6329399-B1 Antifungal amine derivatives and processing for producing the same POLA CHEMICAL INDUSTRIES, INC. (JP) 2001-12-11 US claimed
EP-1020426-A1 AMINE DERIVATIVES AND PROCESS FOR PRODUCING THE SAME POLA CHEMICAL INDUSTRIES, INC. (JP) 2000-07-19 EP claimed
US-6329399-B1 Antifungal amine derivatives and processing for producing the same POLA CHEMICAL INDUSTRIES, INC. (JP) 2001-12-11 US disclosed
EP-1020426-A1 AMINE DERIVATIVES AND PROCESS FOR PRODUCING THE SAME POLA CHEMICAL INDUSTRIES, INC. (JP) 2000-07-19 EP disclosed