SCHEMBL5169656

SCHEMBL5169656

O=C(O)/C=C/c1ccc(N[C@]2(Cc3ccc(F)cc3)CCNC2)nc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.40
P4HTM Q9NXG6 1/20 0.38
GCK P35557 1/20 0.36
AKR1C3 P42330 6/20 0.34
TBXAS1 P24557 2/20 0.34
AKR1C2 P52895 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MITF O75030 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
KLF5 Q13887 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
GSK3B P49841 1/20 0.34
BACE1 P56817 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
DHODH Q02127 1/20 0.33
ESR1 P03372 1/20 0.33
AKR1C4 P17516 1/20 0.33
NOS3 P29474 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5170179 0.91 P4HTM (0.40) HDAC1P4HTMGCKTBXAS1KDM4E
SCHEMBL5170275 0.91 P4HTM (0.40) HDAC1P4HTMGCKTBXAS1KDM4E
SCHEMBL5195209 0.88 SLC6A2 (0.32) HDAC1P4HTMAKR1C3AKR1C2MEN1
SCHEMBL5170448 0.87 THRB (0.45) HDAC1P4HTMGCKAKR1C3AKR1C2
SCHEMBL5169616 0.82 MAPKAPK2 (0.31) HDAC1ALDH1A1SMN1; SMN2
SCHEMBL5168539 0.82 HDAC1 (0.48) HDAC1ALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL5170495 0.81 HDAC1 (0.47) HDAC1ALDH1A1SMN1; SMN2
SCHEMBL5168695 0.80 P4HTM (0.40) HDAC1P4HTMGCKTBXAS1KDM4E
Acetic Acid SCHEMBL5171407 0.79 HDAC1 (0.46) HDAC1ALDH1A1SMN1; SMN2
SCHEMBL5191421 0.78 HDAC3 (0.39) HDAC1P4HTMTBXAS1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1776357-A1 HYDROXYAMIDE COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF HISTONE DEACETYLASE (HDAC) Astellas Pharma Inc. (JP) 2007-04-25 EP disclosed
WO-2006016680-A1 HYDROXYAMIDE COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF HISTONE DEACETYLASE (HDAC) ASTELLAS PHARMA INC. (JP) 2006-02-16 WO disclosed