SCHEMBL5195209

SCHEMBL5195209

O=C(O)/C=C/c1cnc(N[C@]2(Cc3ccc(F)cc3)CCNC2)cn1

nearest known ligand 0.32

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.32
SLC6A4 P31645 2/20 0.32
SLC6A3 Q01959 2/20 0.32
HDAC1 Q13547 2/20 0.32
CYP2D6 P10635 1/20 0.31
KCNH2 Q12809 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
CNR2 P34972 1/20 0.31
AKR1C3 P42330 2/20 0.31
AKR1C4 P17516 1/20 0.31
AKR1C2 P52895 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
P4HTM Q9NXG6 1/20 0.30
CA2 P00918 1/20 0.30
CA5A P35218 1/20 0.30
CA9 Q16790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5169616 0.94 MAPKAPK2 (0.31) SLC6A2SLC6A4SLC6A3HDAC1HDAC3
SCHEMBL5191421 0.91 HDAC3 (0.39) SLC6A2SLC6A4SLC6A3HDAC1CYP2D6
SCHEMBL5170237 0.90 AKR1C3 (0.33) HDAC1HDAC3HDAC2HDAC6AKR1C3
SCHEMBL5195227 0.90 RAB9A (0.32) HDAC1HDAC3HDAC2HDAC6AKR1C3
Hydrochloric Acid SCHEMBL5172809 0.90 HDAC1 (0.36) HDAC1KCNH2HDAC3HDAC2HDAC6
SCHEMBL5171686 0.89 SLC6A2 (0.35) SLC6A2SLC6A3CYP2D6AKR1C3AKR1C2
SCHEMBL5169656 0.88 HDAC1 (0.40) HDAC1AKR1C3AKR1C4AKR1C2MEN1
SCHEMBL5197780 0.85 HDAC3 (0.38) SLC6A2SLC6A4SLC6A3HDAC1CYP2D6
SCHEMBL5171832 0.85 RAB9A (0.31) HDAC1HDAC3HDAC2HDAC6
SCHEMBL5171617 0.85 SLC6A2 (0.34) SLC6A2SLC6A3HDAC1HDAC3HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1776357-A1 HYDROXYAMIDE COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF HISTONE DEACETYLASE (HDAC) Astellas Pharma Inc. (JP) 2007-04-25 EP disclosed
WO-2006016680-A1 HYDROXYAMIDE COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF HISTONE DEACETYLASE (HDAC) ASTELLAS PHARMA INC. (JP) 2006-02-16 WO disclosed