SCHEMBL5169616

SCHEMBL5169616

O=C(O)/C=C/c1cnc(N[C@@]2(Cc3ccc(F)cc3)CCCNC2)cn1

nearest known ligand 0.31

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
HDAC1 Q13547 2/20 0.31
NPC1 O15118 1/20 0.31
CYP1A2 P05177 1/20 0.31
POLB P06746 1/20 0.31
CYP2C19 P33261 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ALDH1A1 P00352 1/20 0.30
ADRB2 P07550 1/20 0.30
HTT P42858 1/20 0.30
HDAC3 O15379 1/20 0.30
HDAC2 Q92769 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5195209 0.94 SLC6A2 (0.32) SLC6A2SLC6A4SLC6A3HDAC1HDAC3
SCHEMBL5197780 0.91 HDAC3 (0.38) SLC6A2SLC6A4SLC6A3HDAC1RAB9A
SCHEMBL5167688 0.91 AKR1C3 (0.32) SLC6A4HDAC1ALDH1A1ADRB2HTT
SCHEMBL5171832 0.91 RAB9A (0.31) HDAC1NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL5191421 0.85 HDAC3 (0.39) SLC6A2SLC6A4SLC6A3HDAC1RAB9A
SCHEMBL5170345 0.85
SCHEMBL5195227 0.85 RAB9A (0.32) HDAC1NPC1RAB9ASMN1; SMN2HDAC3
SCHEMBL5170237 0.85 AKR1C3 (0.33) HDAC1SMN1; SMN2ALDH1A1HDAC3HDAC2
Hydrochloric Acid SCHEMBL5172809 0.84 HDAC1 (0.36) HDAC1HDAC3HDAC2HDAC6
SCHEMBL5169133 0.84 ALDH1A1 (0.35) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1776357-A1 HYDROXYAMIDE COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF HISTONE DEACETYLASE (HDAC) Astellas Pharma Inc. (JP) 2007-04-25 EP disclosed
WO-2006016680-A1 HYDROXYAMIDE COMPOUNDS HAVING ACTIVITY AS INHIBITORS OF HISTONE DEACETYLASE (HDAC) ASTELLAS PHARMA INC. (JP) 2006-02-16 WO disclosed