SCHEMBL5170271

SCHEMBL5170271

O=C(Cl)Oc1ccncc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.54
LMNA P02545 3/20 0.46
CYP1A2 P05177 3/20 0.46
CYP2C19 P33261 3/20 0.46
CYP2C9 P11712 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
CYP19A1 P11511 1/20 0.44
NAPRT Q6XQN6 1/20 0.41
ALDH1A1 P00352 1/20 0.38
MDM2 Q00987 1/20 0.38
NPC1 O15118 2/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2D6 P10635 2/20 0.38
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.37
NFKB1 P19838 2/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37
NPSR1 Q6W5P4 1/20 0.36
KDM4E B2RXH2 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10772752 0.98 HSD17B10 (0.52) HSD17B10LMNACYP1A2CYP2C19CYP2C9
Pyridine SCHEMBL5452272 0.83 CYP19A1 (0.51) HSD17B10LMNACYP1A2CYP2C19CYP2C9
SCHEMBL6924446 0.82 RAB9A (0.46) HSD17B10LMNASMN1; SMN2ALDH1A1KMT2A
SCHEMBL18727667 0.80 HSD17B10 (0.58) HSD17B10LMNACYP1A2CYP2C19CYP2C9
SCHEMBL23355573 0.78 HSD17B10 (0.56) HSD17B10LMNACYP1A2CYP2C19CYP2C9
SCHEMBL380364 0.78 HSD17B10 (0.56) HSD17B10LMNACYP1A2CYP2C19CYP2C9
SCHEMBL1467052 0.76 HSD17B10 (0.54) HSD17B10LMNACYP1A2CYP2C19CYP2C9
SCHEMBL1467050 0.76 HSD17B10 (0.54) HSD17B10LMNACYP1A2CYP2C19CYP2C9
SCHEMBL20412354 0.76 HSD17B10 (0.54) HSD17B10LMNACYP1A2CYP2C19CYP2C9
SCHEMBL27950381 0.76 HSD17B10 (0.54) HSD17B10LMNACYP1A2CYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1776346-B1 1,5-Diphenylpyrazoles MERCK PATENT GMBH (DE) 2013-06-26 EP disclosed
EP-1776346-A1 1,5-DIPHENYLPYRAZOLES Merck Patent GmbH (DE) 2007-04-25 EP disclosed
WO-2006018082-A1 1,5-DIPHENYLPYRAZOLES MERCK PATENT GMBH (DE) 2006-02-23 WO disclosed
EP-0564409-B1 Pyrimidin derivatives and process for their preparation NOVARTIS AG (CH) 2000-01-19 EP disclosed
EP-0564409-A1 Pyrimidin derivatives and process for their preparation CIBA-GEIGY AG (CH) 1993-10-06 EP disclosed
EP-0330927-A2 Pyridine-4-carboxylic-acid anilide BAYER AG (DE) 1989-09-06 EP disclosed
EP-0018533-A1 Substituted pentane (or pentene) carboxylic acids and their derivatives, process for their preparation and their use for the preparation of 3-(arylvinyl)-2,2-dimethyl-cyclopropane-1-carboxylates BAYER AG (DE) 1980-11-12 EP disclosed