SCHEMBL5170782

SCHEMBL5170782

CCS(=O)(=O)c1ccc(C(=O)N[C@@H](C)C(=O)O)c(N)c1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CA2 P00918 9/20 0.50
CA1 P00915 8/20 0.50
CA12 O43570 2/20 0.46
CA9 Q16790 2/20 0.46
FLT1 P17948 1/20 0.39
FLT4 P35916 1/20 0.39
KDR P35968 1/20 0.39
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.38
GAA P10253 1/20 0.37
ADAMTS4 O75173 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2514721 0.78 ALDH1A1 (0.47) CA2ALDH1A1KDM4EPOLBGAA
SCHEMBL5172577 0.77 CA2 (0.70) CA2CA1CA12CA9
SCHEMBL5172574 0.77 CA2 (0.70) CA2CA1CA12CA9
SCHEMBL5173180 0.77 CA2 (0.48) CA2CA1CA12CA9
SCHEMBL23440037 0.72 ALDH1A1 (0.69) CA2CA1ALDH1A1KDM4EGAA
SCHEMBL1533823 0.72 ALDH1A1 (0.69) CA2CA1ALDH1A1KDM4EGAA
SCHEMBL12201410 0.71 USP30 (0.41)
SCHEMBL19332495 0.70 CA2 (0.43) CA2CA1CA12CA9ALDH1A1
SCHEMBL15631042 0.69 ALOX5 (0.49) CA2CA1ALDH1A1
SCHEMBL15631043 0.69 ALOX5 (0.49) CA2CA1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781602-A1 4-SULFONYL-SUBSTITUTED BENZOYLALANINE DERIVATIVES USEFUL AS KYNURENINE-AMINOTRANSFERASE INHIBITORS PELLICCIARI, Roberto (IT) 2007-05-09 EP claimed
WO-2006013085-A1 4-SULFONYL-SUBSTITUTED BENZOYLALANINE DERIVATES USEFUL AS KYNURENINE-AMINOTRANSFERASE INHIBITORS PELLICCIARI ROBERTO (IT) 2006-02-09 WO claimed
EP-1781602-A1 4-SULFONYL-SUBSTITUTED BENZOYLALANINE DERIVATIVES USEFUL AS KYNURENINE-AMINOTRANSFERASE INHIBITORS PELLICCIARI, Roberto (IT) 2007-05-09 EP disclosed
WO-2006013085-A1 4-SULFONYL-SUBSTITUTED BENZOYLALANINE DERIVATES USEFUL AS KYNURENINE-AMINOTRANSFERASE INHIBITORS PELLICCIARI ROBERTO (IT) 2006-02-09 WO disclosed