SCHEMBL5173147

SCHEMBL5173147

CCCC[Si](C)(C)Oc1cccc(C(=O)c2cc(Br)ccc2C(=O)O)c1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AKR1C2 P52895 2/20 0.50
AKR1C1 Q04828 2/20 0.50
POLB P06746 2/20 0.39
KMT2A Q03164 2/20 0.38
MAPT P10636 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38
ALOX12 P18054 1/20 0.38
RECQL P46063 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CYP2C8 P10632 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.37
PLA2G4B P0C869 1/20 0.37
SORT1 Q99523 1/20 0.37
SMPD1 P17405 3/20 0.37
PTPN11 Q06124 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5184110 0.96 AKR1C2 (0.50) AKR1C2AKR1C1POLBKMT2AMAPT
SCHEMBL5155346 0.81 AKR1C2 (0.44) AKR1C2AKR1C1POLBMAPTKDM4E
SCHEMBL4675271 0.78 CYP2C8 (0.59) AKR1C2AKR1C1POLBMAPTKDM4E
SCHEMBL5156418 0.77 AKR1C2 (0.44) AKR1C2AKR1C1POLBMAPTHSD17B10
SCHEMBL4680433 0.73 CYP2C8 (0.59) AKR1C2AKR1C1POLBMAPTKDM4E
SCHEMBL3422610 0.70 MAPT (0.69) POLBKMT2AMAPTKDM4EMEN1
SCHEMBL18529832 0.70 MAOB (0.42) KMT2AKDM4EALDH1A1HPGDHSD17B10
SCHEMBL5188852 0.68 MAPT (0.55) AKR1C2AKR1C1POLBKMT2AMAPT
SCHEMBL6585059 0.67 MGLL (0.43) MAPTKDM4E
SCHEMBL6987433 0.67 LTA4H (0.46) KMT2AMAPTALDH1A1RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740558-A1 BENZOXAZOCINES AND THEIR THERAPEUTIC USE AS MONOAMINE REUPTAKE INHIBITORS Sosei R&D Ltd. (GB) 2007-01-10 EP disclosed
WO-2005103019-A1 BENZOXAZOCINES AND THEIR THERAPEUTIC USE AS MONOAMINE REUPTAKE INHIBITORS SOSEI R&D LTD. (GB) 2005-11-03 WO disclosed