SCHEMBL5175372

SCHEMBL5175372

CCOC(=O)CCCOc1ccc(C[C@H](NC(=O)OCc2ccccc2)C(=O)OC(C)(C)C)cc1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 14/20 0.61
ITGA2B P08514 14/20 0.61
ITGAV P06756 1/20 0.52
LTA4H P09960 3/20 0.50
PTPN1 P18031 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4830419 0.89 ITGB3 (0.70) ITGB3ITGA2BITGAVLTA4H
SCHEMBL7363344 0.85 ITGB3 (0.63) ITGB3ITGA2BITGAV
SCHEMBL8177199 0.84 ITGB3 (0.69) ITGB3ITGA2BLTA4HPTPN1
SCHEMBL8336016 0.84 ITGB3 (0.59) ITGB3ITGA2B
SCHEMBL5175122 0.84 ITGB3 (0.57) ITGB3ITGA2BITGAV
SCHEMBL30149863 0.84 ITGB3 (0.67) ITGB3ITGA2BITGAV
SCHEMBL6287557 0.84 ITGB3 (0.61) ITGB3ITGA2BITGAV
SCHEMBL7412163 0.83 SIRT2 (0.49) ITGB3ITGA2BLTA4H
SCHEMBL8341037 0.83 ITGB3 (0.60) ITGB3ITGA2BITGAV
SCHEMBL19485480 0.83 CTSK (0.62) ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0820991-B1 Cycloalkyl derivatives as bone resorption inhibitors and vitronectin receptor antagonists HOECHST AG (DE) 2007-08-29 EP disclosed
EP-0907637-A1 PHENYLALAMINE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GmbH (DE) 1999-04-14 EP disclosed
EP-0820991-A2 Cycloalkyl derivatives as bone resorption inhibitors and vitronectin receptor antagonists HOECHST AKTIENGESELLSCHAFT (DE) 1998-01-28 EP disclosed
WO-1998000395-A1 PHENYLALAMINE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 1998-01-08 WO disclosed