SCHEMBL5176372

SCHEMBL5176372

CC[C@@H](C)N(C)c1ccc(C#N)c(C#N)c1.CC[C@@H](C)Nc1ccc(C#N)c(C#N)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
TP53 P04637 1/20 0.41
HSP90AA1 P07900 1/20 0.41
CYP3A4 P08684 1/20 0.41
THRB P10828 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
CASP1 P29466 1/20 0.41
HIF1A Q16665 1/20 0.41
HSD17B10 Q99714 1/20 0.41
AR P10275 2/20 0.37
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
PGR P06401 2/20 0.31
NPC1 O15118 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2D6 P10635 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4902159 0.87 AR (0.45) ARMAOAMAOBPGRCYP2C19
SCHEMBL4902166 0.87 AR (0.45) ARMAOAMAOBPGRCYP2C19
SCHEMBL4904892 0.85 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2TDP1L3MBTL1TP53
SCHEMBL4904887 0.85 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2TDP1L3MBTL1TP53
SCHEMBL5074350 0.78 ALDH1A1 (0.64) ALDH1A1SMN1; SMN2TDP1L3MBTL1TP53
SCHEMBL5175006 0.78 ALDH1A1 (0.47) ALDH1A1SMN1; SMN2TDP1L3MBTL1TP53
SCHEMBL4894275 0.74 PGR (0.49) ARPGRCYP2C19
SCHEMBL4894270 0.74 PGR (0.49) ARPGRCYP2C19
SCHEMBL4916336 0.74 MAOA (0.40) ARMAOAMAOBPGRCYP2C19
SCHEMBL4899853 0.74 MAOA (0.40) ARMAOAMAOBPGRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1747193-A1 BENZONITRILE DERIVATIVES TO TREAT MUSCULOSKELETAL FRAILTY Pfizer Products Incorporated (US) 2007-01-31 EP disclosed
WO-2005108351-A1 BENZONITRILE DERIVATIVES TO TREAT MUSCULOSKELETAL FRAILTY PFIZER PRODUCTS INC. (US) 2005-11-17 WO disclosed