SCHEMBL5183162

SCHEMBL5183162

COc1ccc2c(c1)C(C(=O)O)CNC2

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.47
HTR2A P28223 1/20 0.47
HTR2B P41595 1/20 0.47
HSPA1A P0DMV8 1/20 0.43
PTPN7 P35236 1/20 0.43
SIRT1 Q96EB6 1/20 0.43
MTNR1A P48039 4/20 0.40
MTNR1B P49286 4/20 0.39
NQO2 P16083 3/20 0.39
MAPKAPK2 P49137 1/20 0.38
MAPKAPK5 Q8IW41 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA7 P36544 1/20 0.38
CHRNA4 P43681 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30932922 0.87 HTR2A (0.46) HTR2CHTR2AHTR2BMTNR1AMTNR1B
Hydrochloric Acid SCHEMBL5431235 0.86 HTR2A (0.45) HTR2CHTR2AHTR2BMTNR1AMTNR1B
SCHEMBL1520733 0.80 SIRT1 (0.45) SIRT1MTNR1AMTNR1BNQO2
Hydrochloric Acid SCHEMBL17965621 0.78 HTR2C (0.50) HTR2CHTR2AHTR2BCHRNB2CHRNB4
SCHEMBL19748926 0.78 HTR2A (0.42) HTR2CHTR2AHTR2BHSPA1APTPN7
SCHEMBL1842495 0.78 MTNR1A (0.56) MTNR1AMTNR1BNQO2
SCHEMBL30746730 0.78 MTNR1A (0.56) MTNR1AMTNR1BNQO2
SCHEMBL3749345 0.77 HSPA1A (0.51) HTR2CHTR2AHTR2BHSPA1APTPN7
Hydrochloric Acid SCHEMBL9628615 0.77 MTNR1A (0.54) MTNR1AMTNR1BNQO2
SCHEMBL16624059 0.76 HTR2C (0.51) HTR2CHTR2AHTR2BCHRNB2CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1466604-B1 Isoquinoline derivatives, process for their preparation and use thereof in the treatment of melatoninergic system problems SERVIER LAB (FR) 2007-11-07 EP disclosed
EP-1466604-A1 Isoquinoline derivatives, process for their preparation and use thereof in the treatment of melatoninergic system problems Les Laboratoires Servier (FR) 2004-10-13 EP disclosed