SCHEMBL5183222

SCHEMBL5183222

NC(=O)C(=O)NCCS(=O)(=O)O

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.39
SLC6A6 P31641 1/20 0.39
CYP2C19 P33261 1/20 0.39
BLM P54132 1/20 0.39
GAA P10253 1/20 0.37
APP P05067 1/20 0.36
CYP2D6 P10635 1/20 0.35
TGFBR1 P36897 1/20 0.33
PTGS1 P23219 1/20 0.33
PDE4A P27815 1/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA12 O43570 1/20 0.32
CA9 Q16790 1/20 0.32
EPHX2 P34913 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8664606 0.81 LMNA (0.42) LMNASLC6A6CYP2C19BLMAPP
SCHEMBL15808674 0.80 GAA (0.36) GAATGFBR1CA1CA2CA12
SCHEMBL15201198 0.78 GAA (0.52) GAACA1CA2CA12CA9
SCHEMBL31264254 0.77 GAA (0.45) LMNACYP2C19BLMGAATGFBR1
SCHEMBL1404471 0.74 CYP2D6 (0.40) LMNASLC6A6CYP2C19BLMAPP
SCHEMBL28685473 0.74 ALOX15 (0.50) LMNASLC6A6CYP2C19BLMAPP
SCHEMBL33972 0.74 ALOX15 (0.50) LMNASLC6A6CYP2C19BLMAPP
SCHEMBL41304 0.74 TGFBR1 (0.37) LMNASLC6A6CYP2C19BLMCYP2D6
SCHEMBL11693252 0.74 PTGS1 (0.31) LMNASLC6A6CYP2C19BLMCYP2D6
SCHEMBL11690410 0.74 PTGS1 (0.31) LMNASLC6A6CYP2C19BLMCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 70 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102952095-A Synthetic method of 2-carboxylic acid ethyl ester-5-brooethyl thiazole SHENGSHI TAIKE BIOLOG MEDICAL TECHNOLOGY SUZHOU CO LTD 2013-03-06 CN claimed
CN-102666552-B Bicyclic thiazoles as allosteric modulators of the MGLUR5 receptor JANSSEN PHARMACEUTICA NV 2014-11-26 CN disclosed
CN-104086528-A Novel heterocyclic compounds as pesticides BAYER IP GMBH 2014-10-08 CN disclosed
CN-101273042-B Macrocyclic inhibitors of hepatitis C virus TIBOTEC PHARM LTD 2013-11-06 CN disclosed
CN-103130792-A 2-aminothiazoles compound JIANGSU CHIA TAI TIANQING PHAR 2013-06-05 CN disclosed
CN-103140483-A novel heterocyclic compounds as pesticides BAYER CROPSCIENCE AG 2013-06-05 CN disclosed
CN-103130791-A Novel benzamides compound JIANGSU CHIA TAI TIANQING PHAR 2013-06-05 CN disclosed
CN-102952095-A Synthetic method of 2-carboxylic acid ethyl ester-5-brooethyl thiazole SHENGSHI TAIKE BIOLOG MEDICAL TECHNOLOGY SUZHOU CO LTD 2013-03-06 CN disclosed
CN-102947280-A Carboxy-oxazole or thiazole compounds as DGAT-1 inhibitors useful for the treatment of obesity PIRAMAL LIFE SCIENCES LTD 2013-02-27 CN disclosed
CN-101868563-B Base processing agent for metal material and method for processing base for metal material NIHON PARKERIZING 2012-09-12 CN disclosed
CN-1355810-A Prodrugs of thrombin inhibitors BASF AG (DE) 2002-06-26 CN disclosed
CN-1351593-A Substituted polycyclic aryl and heteroaryl pyrymidinones useful as anticoagulants agents PHARMACIA CO (US) 2002-05-29 CN disclosed
CN-1341592-A Proteinase inhibitor SMITHKLINE BEECHEM CORP (US) 2002-03-27 CN disclosed
CN-1341590-A Proteinase inhibitor SMITHKLINE BEECHEM CORP (US) 2002-03-27 CN disclosed
CN-1341593-A Proteinase inhibitor SMITHKLINE BEECHEM CORP (US) 2002-03-27 CN disclosed
CN-1290263-A Arylpiperidine derivatives and use thereof NIHON NOHYAKU CO LTD (JP) 2001-04-04 CN disclosed
CN-1289341-A Thrombin inhibitors BASF AG (DE) 2001-03-28 CN disclosed
CN-1210531-A Dihydrobenzofuran and related compounds useful as anti-inflammatory agents PROCTER & GAMBLE (US) 1999-03-10 CN disclosed
CN-1207095-A Protease inhibitors SMITHKLINE BEECHAM CORP (US) 1999-02-03 CN disclosed
CN-1207102-A 5h,10h-imidazo[1,2-alpha] indeno [1,2-3] pyrazine-4-one derivatives preparation thereof, intermediates thereof and drugs containing same RHONE POULENC RORER SA (FR) 1999-02-03 CN disclosed