SCHEMBL5186000

SCHEMBL5186000

CN(Cc1ccccc1)C(=O)Oc1cccn1C

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
CA12 O43570 1/20 0.47
CA9 Q16790 1/20 0.47
CHRNB2 P17787 1/20 0.46
CHRNB4 P30926 1/20 0.46
CHRNA3 P32297 1/20 0.46
CHRNA4 P43681 1/20 0.46
APOBEC3A P31941 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.44
KMT2A Q03164 3/20 0.44
MEN1 O00255 1/20 0.43
ABHD6 Q9BV23 1/20 0.43
HPGD P15428 1/20 0.42
RIPK1 Q13546 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5187236 0.87 LMNA (0.44) NPC1RAB9AKMT2AMEN1
SCHEMBL5188030 0.82 KMT2A (0.51) SMN1; SMN2KMT2AMEN1
SCHEMBL6273588 0.77 LMNA (0.41) HPGD
SCHEMBL31164812 0.77 NPC1 (0.61) NPC1RAB9ACA12CA9CHRNB2
SCHEMBL2095210 0.76 NPC1 (0.67) NPC1RAB9ACA12CA9CHRNB2
SCHEMBL29020266 0.76 TSHR (0.51) NPC1RAB9ASMN1; SMN2KMT2AHPGD
SCHEMBL5656197 0.75 APOBEC3A (0.55) NPC1RAB9ACA12CA9APOBEC3A
SCHEMBL3882545 0.72 RAB9A (0.39) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL2095207 0.72 NPC1 (0.59) NPC1RAB9ACA12CA9CHRNB2
SCHEMBL6277045 0.71 NPC1 (0.62) NPC1RAB9ACA12CA9SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1751101-A1 SUBSTITUTED 5-AMINOMETHYL-1H-PYRROL-2-CARBXYLIC ACID AMIDES Grünenthal GmbH (DE) 2007-02-14 EP disclosed
WO-2005113497-A1 SUBSTITUTED 5-AMINOMETHYL-1H-PYRROL-2-CARBXYLIC ACID AMIDES Grünenthal GmbH (DE) 2005-12-01 WO disclosed
EP-1581490-A1 SUBSTITUTED 5-AMINOMETHYL-1H-PYRROLE-2-CARBOXAMIDES Grünenthal GmbH (DE) 2005-10-05 EP disclosed
WO-2004058707-A1 SUBSTITUTED 5-AMINOMETHYL-1H-PYRROLE-2-CARBOXAMIDES Grünenthal GmbH (DE) 2004-07-15 WO disclosed