SCHEMBL5186245

SCHEMBL5186245

COc1ccc(-c2coc(N)n2)cc1OC

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.50
ADORA2A P29274 3/20 0.49
KDM4E B2RXH2 5/20 0.48
ALDH1A1 P00352 5/20 0.48
MAPK1 P28482 4/20 0.48
MEN1 O00255 4/20 0.48
KMT2A Q03164 4/20 0.48
SMN1; SMN2 Q16637 4/20 0.48
HSD17B10 Q99714 3/20 0.48
HPGD P15428 3/20 0.48
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
TSHR P16473 2/20 0.48
HTT P42858 2/20 0.48
LTA4H P09960 1/20 0.48
USP2 O75604 1/20 0.48
ATM Q13315 1/20 0.48
AGTR1 P30556 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
ADORA1 P30542 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15100543 0.78 ENPP3 (0.65) KDM4EALDH1A1SMN1; SMN2HSD17B10HPGD
SCHEMBL4530936 0.74 MGAM (0.49) KDM4EALDH1A1MAPK1MEN1KMT2A
SCHEMBL1388381 0.72 DYRK1A (0.66) ADORA2AKDM4EALDH1A1MAPK1MEN1
SCHEMBL427925 0.72 MEN1 (0.75) KDM4EALDH1A1MAPK1MEN1KMT2A
SCHEMBL13210267 0.72 ENPP3 (0.63) KDM4EALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL17144996 0.72 KDM4E (0.65) PDE4AKDM4EALDH1A1MAPK1MEN1
SCHEMBL4831635 0.71 CYP1A2 (0.56) ADORA2AKDM4EALDH1A1MEN1KMT2A
SCHEMBL15100535 0.71 LTA4H (0.55) ADORA2AKDM4EALDH1A1HSD17B10HPGD
SCHEMBL3044785 0.71 KMO (0.55) ADORA2AKDM4EALDH1A1MAPK1MEN1
Bromide SCHEMBL8360766 0.71 NPC1 (0.73) KDM4EALDH1A1MAPK1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1551813-A4 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2007-07-11 EP claimed
EP-1551813-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2005-07-13 EP claimed
WO-2004032882-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2004-04-22 WO claimed