SCHEMBL5186268

SCHEMBL5186268

Cc1cc(-c2cccc(NC(=O)Nc3ccc(Cl)cc3)c2)ncn1.O=C(Nc1ccc(Cl)cc1)Nc1ccc(-c2cccnc2)cc1

nearest known ligand 0.69

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 17/20 0.69
CNR2 P34972 1/20 0.58
MAPT P10636 1/20 0.58
KDR P35968 1/20 0.57
MEN1 O00255 1/20 0.53
RAB9A P51151 1/20 0.53
KMT2A Q03164 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4921639 0.90 CNR1 (0.71) CNR1CNR2MAPT
SCHEMBL30469259 0.83 CNR1 (1.00) CNR1CNR2KDRMEN1RAB9A
SCHEMBL20557904 0.83 CNR1 (1.00) CNR1CNR2KDRMEN1RAB9A
SCHEMBL5186258 0.82 CNR1 (0.47) CNR1CNR2MAPTKDR
SCHEMBL1492983 0.81 PORCN (0.69) CNR1CNR2MAPTKDRRAB9A
SCHEMBL4911349 0.80 CNR1 (0.80) CNR1CNR2MAPTKDRMEN1
SCHEMBL20557632 0.77 CNR1 (1.00) CNR1CNR2MAPT
SCHEMBL30469222 0.77 CNR1 (1.00) CNR1CNR2MAPT
SCHEMBL20557634 0.75 CNR1 (1.00) CNR1CNR2
SCHEMBL30469231 0.75 CNR1 (1.00) CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1786422-A2 ARYL UREA DERIVATIVES FOR TREATING OBESITY Prosidion Limited (GB) 2007-05-23 EP disclosed
WO-2006018662-A2 ARYL UREA DERIVATIVES FOR TREATING OBESITY PROSIDION LIMITED (GB) 2006-02-23 WO disclosed