SCHEMBL5189293

SCHEMBL5189293

CCC(C)(C)C[C@@H](NC(=O)OCc1ccccc1)C(=O)OC

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KYNU Q16719 1/20 0.57
CTSL P07711 3/20 0.56
CTSS P25774 3/20 0.56
CTSB P07858 2/20 0.56
ALDH1A1 P00352 2/20 0.55
ALOX15 P16050 1/20 0.55
CTSK P43235 5/20 0.51
SYK P43405 1/20 0.51
SIRT2 Q8IXJ6 1/20 0.50
SIRT1 Q96EB6 1/20 0.50
SIRT3 Q9NTG7 1/20 0.50
CYP3A4 P08684 1/20 0.49
TSHR P16473 1/20 0.49
MBOAT4 Q96T53 1/20 0.49
TRPM8 Q7Z2W7 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18775057 0.91 CTSS (0.57) KYNUCTSLCTSSCTSBALDH1A1
SCHEMBL18775053 0.91 CTSS (0.57) KYNUCTSLCTSSCTSBALDH1A1
SCHEMBL13863699 0.91 CTSS (0.57) KYNUCTSLCTSSCTSBALDH1A1
SCHEMBL18020341 0.89 CTSS (0.55) KYNUCTSLCTSSCTSBALDH1A1
SCHEMBL15774022 0.89 KYNU (0.56) KYNUCTSLCTSSCTSBALDH1A1
SCHEMBL3044553 0.88 CTSS (0.70) KYNUCTSLCTSSCTSBALDH1A1
SCHEMBL4837883 0.88 KYNU (0.55) KYNUCTSLCTSSCTSBALDH1A1
SCHEMBL4837891 0.88 KYNU (0.55) KYNUCTSLCTSSCTSBALDH1A1
SCHEMBL16346611 0.87 KYNU (0.59) KYNUCTSLCTSSCTSBALDH1A1
SCHEMBL1198823 0.86 KYNU (0.56) KYNUCTSLCTSSCTSBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7531507-B2 Acylated nonadepsipeptides containing pyridyl alanine residues AICURIS GMBH & CO. KG (DE) 2009-05-12 US disclosed
US-7531507-B2 Acylated nonadepsipeptides containing pyridyl alanine residues AICURIS GMBH & CO. KG (DE) 2009-05-12 US disclosed
EP-1807443-A1 ACYLATED NONADEPSIPEPTIDES USED AS LYSOBACTIN DERIVATIVES AiCuris GmbH & Co. KG (DE) 2007-07-18 EP disclosed
WO-2006048139-A1 ACYLATED NONADEPSIPEPTIDES USED AS LYSOBACTIN DERIVATIVES AICURIS GMBH & CO. KG (DE) 2006-05-11 WO disclosed