SCHEMBL5190834

SCHEMBL5190834

NC(=O)CC1CN(C(=O)Nc2ccc(Cl)c(Cl)c2)CCN1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 13/20 0.58
KCNH2 Q12809 13/20 0.58
NPC1 O15118 2/20 0.52
RAB9A P51151 2/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
CCR5 P51681 1/20 0.52
LMNA P02545 3/20 0.51
TP53 P04637 2/20 0.51
MAPT P10636 2/20 0.51
HPGD P15428 1/20 0.48
TSHR P16473 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C19 P33261 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5193648 0.82 POLB (0.53) NPC1RAB9ATP53MAPTHPGD
SCHEMBL5191591 0.80 TP53 (0.53) CCR2KCNH2NPC1RAB9AMEN1
SCHEMBL5193199 0.80 MAPT (0.55) CCR2NPC1RAB9AMEN1KMT2A
SCHEMBL5210355 0.78 CCR2 (0.50) CCR2KCNH2NPC1RAB9AMEN1
SCHEMBL5193560 0.78 CCR2 (0.48) CCR2KCNH2MEN1KMT2ALMNA
SCHEMBL5193950 0.76 CCR2 (0.46) CCR2KCNH2MEN1KMT2ACCR5
SCHEMBL5192584 0.76 CCR3 (0.51) CCR2KCNH2MEN1KMT2ACCR5
SCHEMBL5190802 0.76 CCR2 (0.47) CCR2KCNH2MEN1KMT2ACCR5
SCHEMBL1944478 0.75 NPC1 (0.73) CCR2KCNH2NPC1RAB9AMEN1
Hydrochloric Acid SCHEMBL1943329 0.74 NPC1 (0.71) CCR2KCNH2NPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP disclosed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP disclosed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO disclosed