SCHEMBL5191591

SCHEMBL5191591

Cc1ccc(CNC(=O)CC2CN(C(=O)Nc3ccc(Cl)c(Cl)c3)CCN2)cc1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.53
MAPT P10636 3/20 0.53
LMNA P02545 2/20 0.53
CCR2 P41597 9/20 0.52
KCNH2 Q12809 9/20 0.52
CCR5 P51681 1/20 0.47
PREP P48147 1/20 0.45
POLB P06746 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
PAX8 Q06710 2/20 0.43
MEN1 O00255 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
KMT2A Q03164 1/20 0.43
TDP1 Q9NUW8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5210355 0.90 CCR2 (0.50) TP53MAPTLMNACCR2KCNH2
SCHEMBL5192584 0.85 CCR3 (0.51) LMNACCR2KCNH2CCR5SMN1; SMN2
SCHEMBL5193739 0.84 PKM (0.56) MAPTLMNAPOLBSMN1; SMN2MEN1
SCHEMBL5193560 0.81 CCR2 (0.48) MAPTLMNACCR2KCNH2MEN1
SCHEMBL5190802 0.81 CCR2 (0.47) TP53MAPTLMNACCR2KCNH2
SCHEMBL5190834 0.80 CCR2 (0.58) TP53MAPTLMNACCR2KCNH2
SCHEMBL5193432 0.80 MAPT (0.50) TP53MAPTSMN1; SMN2MEN1RAB9A
SCHEMBL5191220 0.80 FAAH (0.51) TP53MAPTLMNAPOLBSMN1; SMN2
SCHEMBL5193950 0.79 CCR2 (0.46) CCR2KCNH2CCR5MEN1KMT2A
SCHEMBL5194091 0.76 FAAH (0.53) SMN1; SMN2MEN1NPC1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP disclosed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP disclosed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO disclosed