SCHEMBL5191850

SCHEMBL5191850

COc1ccc(CN2CCNC(CC(N)=O)C2)cc1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.49
KDM4E B2RXH2 1/20 0.47
OPRM1 P35372 1/20 0.45
OPRK1 P41145 1/20 0.45
SIGMAR1 Q99720 2/20 0.44
POLB P06746 1/20 0.44
PKM P14618 1/20 0.44
SLC18A3 Q16572 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43
DRD4 P21917 1/20 0.43
MLNR O43193 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10674002 0.84 LTA4H (0.54) LTA4HKDM4ESIGMAR1PKM
SCHEMBL5191015 0.81 SMN1; SMN2 (0.56) SIGMAR1SMN1; SMN2
SCHEMBL28046102 0.79 KDM4E (0.47) KDM4ESIGMAR1POLBPKMSLC18A3
SCHEMBL7063658 0.79 NPY2R (0.41) KDM4EPOLBSMN1; SMN2
SCHEMBL4287551 0.78 LTA4H (0.63) LTA4HSIGMAR1SMN1; SMN2DRD4
SCHEMBL12520647 0.78 LTA4H (0.63) LTA4HSIGMAR1SMN1; SMN2DRD4
SCHEMBL5192443 0.77 ALDH1A1 (0.48) KDM4EPOLBSMN1; SMN2
SCHEMBL6076846 0.76 MLNR (0.49) LTA4HMLNR
SCHEMBL5193199 0.76 MAPT (0.55) SMN1; SMN2
SCHEMBL691646 0.76 LTA4H (0.54) LTA4HSIGMAR1PKMDRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP disclosed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP disclosed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO disclosed