SCHEMBL5193196

SCHEMBL5193196

O=C(N[C@H](C(=O)O)C1CCCCC1)c1ccc(F)cc1[N+](=O)[O-]

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PYGL P06737 14/20 0.55
CTSL P07711 1/20 0.43
EPHX2 P34913 1/20 0.42
CYP2C9 P11712 1/20 0.41
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5193186 1.00 PYGL (0.55) PYGLCTSLEPHX2CYP2C9CNR1
SCHEMBL5196786 0.99 PYGL (0.53) PYGLCTSLEPHX2CYP2C9
SCHEMBL5196793 0.99 PYGL (0.53) PYGLCTSLEPHX2CYP2C9
SCHEMBL5193891 0.89 PYGL (0.52) PYGLCYP2C9
SCHEMBL5195668 0.88 PYGL (0.46) PYGLCYP2C9CNR1CNR2
SCHEMBL5195537 0.86 ALDH1A1 (0.49) PYGL
SCHEMBL5195581 0.86 ALDH1A1 (0.49) PYGL
SCHEMBL5194468 0.86 PYGL (0.43) PYGLCYP2C9CNR1CNR2
SCHEMBL5197192 0.86 PYGL (0.43) PYGLCYP2C9CNR1CNR2
SCHEMBL5195548 0.86 ALDH1A1 (0.49) PYGL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1812383-A1 GLYCOGEN PHOSPHORYLASE INHIBITOR COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF Smithkline Beecham Corporation (US) 2007-08-01 EP disclosed
WO-2006052722-A1 GLYCOGEN PHOSPHORYLASE INHIBITOR COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF SMITHKLINE BEECHAM CORPORATION (US) 2006-05-18 WO disclosed