SCHEMBL5195352

SCHEMBL5195352

COc1ccc(CCNC(=O)CC2CCCCN2)cc1

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.58
SMN1; SMN2 Q16637 1/20 0.52
HPGD P15428 2/20 0.52
MAPT P10636 2/20 0.52
POLB P06746 2/20 0.52
KDM4E B2RXH2 1/20 0.52
MAPK1 P28482 1/20 0.52
HSD17B10 Q99714 1/20 0.52
EPHX2 P34913 1/20 0.50
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA9 Q16790 1/20 0.50
PTPN1 P18031 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5195710 0.89 ALDH1A1 (0.58) ALDH1A1SMN1; SMN2POLBEPHX2CA12
SCHEMBL5193856 0.86 KDM4E (0.55) ALDH1A1POLBKDM4ECA1CA2
SCHEMBL5191195 0.85 MEN1 (0.59) ALDH1A1HPGDMAPTKDM4EHSD17B10
SCHEMBL5193954 0.84 EPHX2 (0.50) POLBEPHX2
SCHEMBL5190605 0.79 ALDH1A1 (0.54) ALDH1A1SMN1; SMN2HPGDMAPTPOLB
SCHEMBL5190612 0.78 KMT2A (0.58) ALDH1A1SMN1; SMN2HPGDPOLBKDM4E
SCHEMBL5195925 0.77 KMT2A (0.58) ALDH1A1HPGDPOLBKDM4E
SCHEMBL21540797 0.77 HTR2C (0.57) ALDH1A1SMN1; SMN2POLBKDM4E
SCHEMBL5194022 0.76 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2HPGDMAPTPOLB
SCHEMBL12773610 0.76 SMN1; SMN2 (0.75) ALDH1A1SMN1; SMN2HPGDPOLBCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP disclosed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP disclosed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO disclosed