SCHEMBL5197682

SCHEMBL5197682

C=CCC(N)CC(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
CYP2D6 P10635 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.34
GRIK1 P39086 2/20 0.33
GRIK2 Q13002 2/20 0.33
USP2 O75604 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
CTSK P43235 2/20 0.31
CYP3A4 P08684 1/20 0.31
TSHR P16473 1/20 0.31
CYP2C19 P33261 1/20 0.31
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22960731 0.83 GRIK1 (0.32) GRIK1GRIK2
SCHEMBL31301962 0.82 CYP2D6 (0.44) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL28507298 0.80 HDAC3 (0.44) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL14524872 0.80 HDAC3 (0.44) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL7275993 0.79 ALDH1A1 (0.44) GRIK1GRIK2TSHRALDH1A1LMNA
Hydrochloric Acid SCHEMBL6972258 0.78 LMNA (0.43) GRIK1GRIK2TSHRALDH1A1LMNA
SCHEMBL28073409 0.78 ALDH1A1 (0.41) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL2189972 0.77 GRIK1 (0.43) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL2189967 0.77 GRIK1 (0.43) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL7052679 0.77 GRIK1 (0.43) HDAC3HDAC1HDAC2HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1814852-A2 HYDROXYBENZOATE SALTS OF METANICOTINE COMPOUNDS Targacept, Inc. (US) 2007-08-08 EP disclosed
EP-1814853-A2 HYDROXYBENZOATE SALTS OF METANICOTINE COMPOUNDS Targacept, Inc. (US) 2007-08-08 EP disclosed
WO-2006053082-A2 HYDROXYBENZOATE SALTS OF METANICOTINE COMPOUNDS TARGACEPT, INC. (US) 2006-05-18 WO disclosed
WO-2006053039-A2 HYDROXYBENZOATE SALTS OF METANICOTINE COMPOUNDS TARGACEPT, INC. (US) 2006-05-18 WO disclosed