SCHEMBL5199072

SCHEMBL5199072

CN1CCN(c2ccc(Nc3ncco3)cc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 4/20 0.54
ADRA2C P18825 4/20 0.54
ADRA2B P18089 3/20 0.54
RAD52 P43351 1/20 0.50
GFER P55789 1/20 0.50
KDM1A O60341 1/20 0.48
GLA P06280 1/20 0.48
SLC2A1 P11166 1/20 0.48
RECQL P46063 1/20 0.48
BLM P54132 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
MAPKAPK2 P49137 6/20 0.47
JAK2 O60674 2/20 0.47
EGFR P00533 1/20 0.47
JAK3 P52333 1/20 0.47
CCNE1 P24864 1/20 0.47
CDK2 P24941 1/20 0.47
ADRB2 P07550 1/20 0.46
CHRM2 P08172 1/20 0.46
CHRM1 P11229 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5199413 0.85 CD274 (0.46) ADRA2AADRA2CADRA2BGFERTDP1
SCHEMBL5200210 0.85 PLK4 (0.53) KDM1ASLC2A1JAK2
SCHEMBL5200215 0.80 JAK2 (0.54) JAK2EGFRJAK3CDK2TNIK
SCHEMBL30854951 0.80 NCF1 (0.50) KDM1ATDP1JAK2JAK3HTR6
SCHEMBL4078840 0.76 EGFR (0.60) ADRA2AADRA2CADRA2BKDM1AGLA
SCHEMBL30925347 0.74 ADRA2C (0.50) ADRA2AADRA2CADRA2BRAD52GFER
SCHEMBL27020409 0.73 EGFR (0.64) ADRA2AADRA2CTDP1JAK2EGFR
SCHEMBL30306480 0.72 EGFR (0.60) ADRA2AADRA2CADRA2BJAK2EGFR
SCHEMBL12325149 0.72 BRD4 (0.64) RAD52GFERJAK2EGFRJAK3
SCHEMBL6968717 0.72 BRD4 (0.61) ADRA2AADRA2CADRA2BRAD52GFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1551813-A4 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2007-07-11 EP disclosed
EP-1551813-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2005-07-13 EP disclosed
WO-2004032882-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2004-04-22 WO disclosed