SCHEMBL5200513

SCHEMBL5200513

COC(=O)c1ccc(CCCNC(=O)OC(C)(C)C)cc1O

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA1 P00915 10/20 0.47
CA2 P00918 10/20 0.47
MTNR1A P48039 1/20 0.46
MTNR1B P49286 1/20 0.46
CA12 O43570 5/20 0.44
CA9 Q16790 5/20 0.44
CA7 P43166 1/20 0.44
PDK2 Q15119 1/20 0.44
PDK4 Q16654 1/20 0.44
CA14 Q9ULX7 1/20 0.44
GAA P10253 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
NQO2 P16083 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
PPARA Q07869 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8003356 0.93 CA2 (0.48) CA1CA2CA12CA9CA7
SCHEMBL7398526 0.82 CA12 (0.59) CA1CA2CA12CA9CA7
SCHEMBL14524170 0.81 CA1 (0.42) CA1CA2CA12CA9TDP1
SCHEMBL21221559 0.81 CYP4A11 (0.57) CA1CA2GAATDP1SIGMAR1
SCHEMBL5961112 0.80 CA12 (0.42) CA1CA2MTNR1AMTNR1BCA12
SCHEMBL6422546 0.79 PPARA (0.43) CA1CA2MTNR1AMTNR1BCA12
SCHEMBL31747308 0.79 CYP4F2 (0.60) MTNR1AMTNR1BNQO2SIGMAR1MEN1
SCHEMBL5725025 0.79 CYP4F2 (0.60) MTNR1AMTNR1BNQO2SIGMAR1MEN1
SCHEMBL22996206 0.79 CA1 (0.54) CA1CA2CA12CA9GAA
SCHEMBL7465537 0.79 ESRRG (0.58) CA1CA2CA12CA9GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1817287-A1 AROMATIC ETHER DERIVATIVES USEFUL AS THROMBIN INHIBITORS Eli Lilly and Company (US) 2007-08-15 EP disclosed
WO-2006057845-A1 AROMATIC ETHER DERIVATIVES USEFUL AS THROMBIN INHIBITORS ELI LILLY AND COMPANY (US) 2006-06-01 WO disclosed