SCHEMBL8003356

SCHEMBL8003356

COC(=O)c1ccc(CCNC(=O)OC(C)(C)C)cc1O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 6/20 0.48
CA1 P00915 5/20 0.48
CA12 O43570 2/20 0.47
CA9 Q16790 2/20 0.47
CA7 P43166 1/20 0.47
PDK2 Q15119 1/20 0.47
PDK4 Q16654 1/20 0.47
CA14 Q9ULX7 1/20 0.47
MAPT P10636 3/20 0.46
KDM4E B2RXH2 2/20 0.46
ALDH1A1 P00352 2/20 0.46
HPGD P15428 2/20 0.46
HSD17B10 Q99714 2/20 0.46
LMNA P02545 2/20 0.46
PTGS1 P23219 1/20 0.46
BLM P54132 1/20 0.46
HIF1A Q16665 1/20 0.46
NQO2 P16083 1/20 0.46
NAMPT P43490 1/20 0.45
GAA P10253 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5200513 0.93 CA1 (0.47) CA2CA1CA12CA9CA7
SCHEMBL30423117 0.85 MAPT (0.63) CA2CA1MAPTKDM4EALDH1A1
SCHEMBL233765 0.85 MAPT (0.63) CA2CA1MAPTKDM4EALDH1A1
SCHEMBL19026301 0.84 CA1 (0.45) CA2CA1MAPTKDM4ELMNA
SCHEMBL8383176 0.83 CYP1A2 (0.51) CA2CA1CA12CA9MAPT
SCHEMBL29998779 0.81 MTNR1A (0.59) CA2CA1CA12CA9LMNA
SCHEMBL69181 0.81 MTNR1A (0.59) CA2CA1CA12CA9LMNA
SCHEMBL27438451 0.81 CA2 (0.49) CA2CA1CA12CA9MAPT
SCHEMBL3698093 0.80 ESRRG (0.53) CA2CA1CA12CA9MAPT
SCHEMBL3706599 0.80 CA12 (0.58) CA2CA1CA12CA9CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000027790-A1 MUTILIN COMPOUNDS SMITHKLINE BEECHAM P.L.C. (GB) 2000-05-18 WO disclosed