SCHEMBL5961112

SCHEMBL5961112

COC(=O)c1ccc(CCCCNCC(=O)OC(C)(C)C)cc1O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42
PDK2 Q15119 1/20 0.42
PDK4 Q16654 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42
PPARA Q07869 1/20 0.41
GAA P10253 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.38
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
KMT2A Q03164 1/20 0.37
HSD17B10 Q99714 1/20 0.37
XDH P47989 1/20 0.37
MYC P01106 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6422546 0.99 PPARA (0.43) CA12CA1CA2CA7PDK2
SCHEMBL5200513 0.80 CA1 (0.47) CA12CA1CA2CA7PDK2
SCHEMBL8003356 0.77 CA2 (0.48) CA12CA1CA2CA7PDK2
SCHEMBL4601057 0.76 CYP4A11 (0.60) CA12CA1CA2CA7PDK2
SCHEMBL5961082 0.76 CA12 (0.43) CA12CA1CA2CA7PDK2
SCHEMBL5961083 0.76 CA12 (0.43) CA12CA1CA2CA7PDK2
SCHEMBL20503308 0.75 PPARA (0.71) CA12CA1CA2CA7PDK2
SCHEMBL31586510 0.75 PPARA (0.71) CA12CA1CA2CA7PDK2
SCHEMBL29102441 0.74 PPARA (0.66) PPARA
SCHEMBL6289030 0.73 CA12 (0.48) CA12CA1CA2CA7PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39088-E1 Amide compounds and use of the same JAPAN TOBACCO, INC. (JP) 2006-05-02 US disclosed
EP-0849256-B1 AMIDE COMPOUNDS AND USE OF THE SAME JAPAN TOBACCO INC (JP) 2005-06-08 EP disclosed
EP-1304322-A2 Carboxylic acid compound and use thereof Japan Tobacco Inc. (JP) 2003-04-23 EP disclosed
US-6420561-B1 Amide compounds and use thereof JAPAN TOBACCO INC. (JP) 2002-07-16 US disclosed
US-6174887-B1 Amide compounds and use of the same JAPAN TOBACCO INC. (JP) 2001-01-16 US disclosed
EP-0849256-A1 AMIDE COMPOUNDS AND USE OF THE SAME Japan Tobacco Inc. (JP) 1998-06-24 EP disclosed