SCHEMBL5200725

SCHEMBL5200725

CN1CCN(c2ccc(-c3nc4cc(NC(=O)c5ccccc5Cl)ccc4[nH]3)cc2)CC1

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NR2E3 Q9Y5X4 17/20 0.59
MT-CO2 P00403 1/20 0.53
RAB9A P51151 2/20 0.52
NPC1 O15118 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4481398 0.87 MT-CO2 (0.50) NR2E3MT-CO2RAB9ANPC1
SCHEMBL6120531 0.85 NPC1 (0.60) RAB9ANPC1
SCHEMBL6126326 0.85 ACHE (0.58) RAB9ANPC1
SCHEMBL1664926 0.82 ACHE (0.54) RAB9ANPC1
SCHEMBL5190803 0.81 NR2E3 (0.65) NR2E3RAB9ANPC1
SCHEMBL8769900 0.81 ACHE (0.54) RAB9ANPC1
SCHEMBL6126388 0.81 ACHE (0.54) RAB9ANPC1
SCHEMBL5205370 0.81 ALDH1A1 (0.48)
SCHEMBL1664044 0.80 NPC1 (0.53) NR2E3RAB9ANPC1
SCHEMBL17072263 0.80 FGFR1 (0.59) RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833829-A2 BENZAMIDE SUBSTITUTED IMIDAZO- AND PYRROLO-PYRIDINES AS PROTEIN KINASE INHIBITORS F. Hoffmann-Roche AG (CH) 2007-09-19 EP disclosed
WO-2006066913-A2 BENZAMIDE SUBSTITUTED IMIDAZO- AND PYROLO-PYRIDINES AS PROTEIN KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2006-06-29 WO disclosed