SCHEMBL5200810

SCHEMBL5200810

CS(=O)(=O)Nc1cccc(CC2=NCCN2)c1Cl

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 5/20 0.51
ADRA1A P35348 12/20 0.47
ADRA2C P18825 11/20 0.47
ADRA2A P08913 6/20 0.47
ADRA2B P18089 3/20 0.47
MAPK1 P28482 2/20 0.47
LMNA P02545 1/20 0.47
HTR1A P08908 1/20 0.47
CYP2D6 P10635 1/20 0.47
MAPT P10636 1/20 0.47
OPRM1 P35372 1/20 0.47
NISCH Q9Y2I1 1/20 0.47
ADRA1D P25100 9/20 0.46
ADRA1B P35368 9/20 0.46
HTR1D P28221 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5203153 0.99 TAAR1 (0.50) TAAR1ADRA1AADRA2CADRA2AADRA2B
SCHEMBL5200657 0.86 TAAR1 (0.52) TAAR1ADRA1AADRA2CADRA2AADRA2B
Hydrochloric Acid SCHEMBL5203075 0.85 TAAR1 (0.51) TAAR1ADRA1AADRA2CADRA2AADRA2B
SCHEMBL5203304 0.84 TAAR1 (0.60) TAAR1ADRA1AADRA2CADRA2AADRA2B
SCHEMBL4986530 0.84 ADRA1A (0.50) TAAR1ADRA1AADRA2CADRA2AADRA2B
SCHEMBL14092049 0.83 HTR1D (0.49) TAAR1ADRA1AADRA2CADRA2AADRA2B
SCHEMBL2387364 0.83 ADRA1A (0.45) TAAR1ADRA1AADRA2CADRA2AADRA2B
Hydrochloric Acid SCHEMBL5203467 0.82 TAAR1 (0.48) TAAR1ADRA1AADRA2CADRA2AADRA2B
Hydrochloric Acid SCHEMBL3726001 0.82 ADRA1A (0.44) TAAR1ADRA1AADRA2CADRA2AADRA2B
SCHEMBL5204270 0.82 TAAR1 (0.48) TAAR1ADRA1AADRA2CADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0887346-B1 N-Phenyl-alkylsulfonamide derivatives, their preparation and their use as alpha1A/1L adrenoceptor agonists HOFFMANN LA ROCHE (CH) 2007-12-12 EP disclosed