SCHEMBL5201503

SCHEMBL5201503

c1ccc(-n2ccc3nncc-3c2)cc1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 6/20 0.45
GABRB3 P28472 6/20 0.45
GABRA5 P31644 6/20 0.45
GABRA3 P34903 6/20 0.45
GABRA1 P14867 4/20 0.43
HPGD P15428 1/20 0.41
COMT P21964 3/20 0.40
CYP3A4 P08684 1/20 0.36
GRM5 P41594 1/20 0.35
DRD4 P21917 2/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
NLRP3 Q96P20 1/20 0.33
KMT2A Q03164 2/20 0.33
P2RX7 Q99572 1/20 0.33
MEN1 O00255 1/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16212535 0.71 GABRG2 (0.35) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL5201498 0.70 NPC1 (0.41) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL14007395 0.70 COMT (0.48) HPGDCOMTCYP3A4GRM5DRD4
SCHEMBL17267004 0.70 COMT (0.48) HPGDCOMTCYP3A4GRM5DRD4
SCHEMBL3227703 0.69 GABRG2 (0.64) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL5785754 0.68 NPC1 (0.50) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL790464 0.67 SCN4A (0.31) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL6110315 0.64 GABRG2 (0.38) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL9466146 0.63 HPGD (0.40) HPGDCOMTCYP3A4GRM5DRD4
SCHEMBL28092437 0.63 CYP1A2 (0.52) HPGDCOMTCYP3A4DRD4NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1744735-A2 METHOD OF TREATMENT OF MYOCARDIAL INFARCTION The Scripps Research Institute (US) 2007-01-24 EP disclosed
WO-2005089366-A2 METHOD OF TREATMENT OF MYOCARDIAL INFARCTION THE SCRIPPS RESEARCH INSTITUTE (US) 2005-09-29 WO disclosed