SCHEMBL5201588

SCHEMBL5201588

N#Cc1c(-c2ccccc2)[nH]c2ccccc12

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.68
DYRK1A Q13627 2/20 0.63
PDE9A O76083 3/20 0.58
ESR1 P03372 3/20 0.55
ESR2 Q92731 3/20 0.55
MAOA P21397 1/20 0.49
MAOB P27338 1/20 0.49
NPSR1 Q6W5P4 1/20 0.46
PDE10A Q9Y233 3/20 0.46
DHODH Q02127 1/20 0.46
PDE1C Q14123 1/20 0.45
IMPDH2 P12268 1/20 0.44
HSD11B1 P28845 1/20 0.44
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
MAPT P10636 1/20 0.44
KMT2A Q03164 1/20 0.44
GPR3 P46089 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11339067 0.87 CYP19A1 (0.53) CYP19A1DYRK1APDE9AESR1ESR2
SCHEMBL28819042 0.86 ESR2 (0.60) CYP19A1DYRK1APDE9AESR1ESR2
SCHEMBL16382906 0.82 HPGD (0.53) CYP19A1DYRK1APDE9AMAOAMAOB
SCHEMBL1606265 0.82 CYP11B2 (0.61) CYP19A1DYRK1APDE9APDE10ADHODH
SCHEMBL28842406 0.82 DYRK1A (0.49) CYP19A1DYRK1APDE9APDE10ADHODH
SCHEMBL15058476 0.78 HTR1A (0.55) DYRK1AIMPDH2ALDH1A1KDM4EMEN1
SCHEMBL10097356 0.78 ALDH1A1 (0.53) DYRK1AMAOAMAOBNPSR1IMPDH2
SCHEMBL16382889 0.78 DYRK1A (0.49) CYP19A1DYRK1APDE9AMAOAMAOB
SCHEMBL28842633 0.78 DYRK1A (0.46) CYP19A1DYRK1APDE9AMAOAMAOB
SCHEMBL25929859 0.78 PDE9A (0.47) CYP19A1DYRK1APDE9APDE1CIMPDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106631982-A Method for synthesizing amino-substituted carbazole compound 河南师范大学 2017-05-10 CN disclosed
WO-2017031276-A1 METHODS OF PROVIDING NEUROPROTECTIVE THERAPY RELATED TO ADMINISTERING AN ESTROGEN RECEPTOR BETA LIGAND THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2017-02-23 WO disclosed
EP-1829872-B1 PROCESSES FOR PRODUCTION OF INDOLE COMPOUNDS NISSAN CHEMICAL IND LTD (JP) 2015-07-29 EP disclosed
EP-1829872-A1 PROCESSES FOR PRODUCTION OF INDOLE COMPOUNDS Nissan Chemical Industries, Ltd. (JP) 2007-09-05 EP disclosed