SCHEMBL5201844

SCHEMBL5201844

O=c1ccc2c[c]c(CO)cc2o1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 14/20 0.50
CA12 O43570 12/20 0.50
CA7 P43166 6/20 0.50
CA4 P22748 4/20 0.50
CA5A P35218 4/20 0.50
CA14 Q9ULX7 4/20 0.50
CA5B Q9Y2D0 3/20 0.50
CA3 P07451 3/20 0.50
CA6 P23280 3/20 0.50
CA2 P00918 2/20 0.50
KDM4E B2RXH2 7/20 0.47
CA1 P00915 7/20 0.47
MCL1 Q07820 6/20 0.47
GLA P06280 6/20 0.47
HSD17B10 Q99714 5/20 0.47
ALDH1A1 P00352 5/20 0.47
AKR1B1 P15121 5/20 0.47
GAA P10253 5/20 0.47
HPGD P15428 4/20 0.47
CASP1 P29466 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1490920 0.77 CA9 (0.56) CA9CA12CA7CA4CA5A
SCHEMBL5204008 0.74 ALDH1A1 (0.50) CA9CA12CA7CA4CA5A
SCHEMBL5200967 0.74 CA12 (0.47) CA9CA12CA7CA4CA5A
SCHEMBL5203277 0.74 CA9 (0.47) CA9CA12CA7CA4CA5A
SCHEMBL15267536 0.73 CA9 (0.62) CA9CA12CA7CA4CA5A
SCHEMBL29603488 0.72 CA12 (0.77) CA9CA12CA7CA4CA5A
SCHEMBL3326190 0.72 CA12 (0.77) CA9CA12CA7CA4CA5A
SCHEMBL5202137 0.70 PGR (0.47) CA9CA12CA7CA4CA5A
SCHEMBL15171953 0.68 CA9 (0.68) CA9CA12CA7CA4CA5A
SCHEMBL10350668 0.67 CA12 (1.00) CA9CA12CA7CA4CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0998474-B1 PIPERAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2007-02-07 EP disclosed
EP-0998474-A1 PIPERAZINE DERIVATIVES MERCK PATENT GmbH (DE) 2000-05-10 EP disclosed
WO-1999003855-A1 PIPERAZINE DERIVATIVES MERCK PATENT GMBH (DE) 1999-01-28 WO disclosed