SCHEMBL5204008

SCHEMBL5204008

Cc1[c]cc2ccc(=O)oc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.50
MCL1 Q07820 7/20 0.49
KMT2A Q03164 3/20 0.47
CA9 Q16790 12/20 0.47
CA12 O43570 11/20 0.47
KDM4E B2RXH2 7/20 0.47
CA1 P00915 7/20 0.47
CA7 P43166 6/20 0.47
HSD17B10 Q99714 5/20 0.47
AKR1B1 P15121 5/20 0.47
HPGD P15428 4/20 0.47
CA4 P22748 4/20 0.47
CA6 P23280 4/20 0.47
CA14 Q9ULX7 4/20 0.47
CA5A P35218 3/20 0.47
CA3 P07451 3/20 0.47
GAA P10253 5/20 0.47
GLA P06280 5/20 0.47
CASP1 P29466 3/20 0.47
CASP7 P55210 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3369222 0.85 ALDH1A1 (0.55) ALDH1A1MCL1KMT2ACA9CA12
SCHEMBL5203277 0.78 CA9 (0.47) ALDH1A1MCL1KMT2ACA9CA12
SCHEMBL5200967 0.78 CA12 (0.47) ALDH1A1MCL1KMT2ACA9CA12
SCHEMBL1490920 0.78 CA9 (0.56) ALDH1A1MCL1KMT2ACA9CA12
SCHEMBL5202137 0.77 PGR (0.47) ALDH1A1MCL1KMT2ACA9CA12
SCHEMBL5201844 0.74 CA9 (0.50) ALDH1A1MCL1KMT2ACA9CA12
SCHEMBL76393 0.72 ALDH1A1 (0.74) ALDH1A1MCL1KMT2ACA9CA12
SCHEMBL8036025 0.72 ALDH1A1 (0.62) ALDH1A1MCL1KMT2ACA9CA12
SCHEMBL4471575 0.71 CYP2A6 (0.36) KDM4EHSD17B10ACHECYP3A4CYP2A6
SCHEMBL11194490 0.68 GAA (0.64) ALDH1A1MCL1KMT2ACA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0998474-B1 PIPERAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2007-02-07 EP disclosed
EP-0998474-A1 PIPERAZINE DERIVATIVES MERCK PATENT GmbH (DE) 2000-05-10 EP disclosed
WO-1999003855-A1 PIPERAZINE DERIVATIVES MERCK PATENT GMBH (DE) 1999-01-28 WO disclosed