SCHEMBL5201877

SCHEMBL5201877

O=CCc1csc(-c2ncc[nH]2)n1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 1/20 0.35
SCN9A Q15858 1/20 0.35
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
NISCH Q9Y2I1 2/20 0.32
MTOR P42345 1/20 0.32
ADK P55263 1/20 0.32
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
BRD4 O60885 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27905839 0.72 SCN9A (0.48) SCN9AADORA2AADORA1NISCHMTOR
SCHEMBL30641564 0.70 PDE10A (0.46) SCN9AADORA2AADORA1NISCHMTOR
SCHEMBL27609155 0.69 ALDH1A1 (0.46) NISCHMTORADKKDM4EALDH1A1
SCHEMBL30785478 0.68 KDM4E (0.54) KDM4E
SCHEMBL5200449 0.68 BRD4 (0.37) ADORA2AADORA1NISCHMTORADK
SCHEMBL3065277 0.67 PDE4A (0.42) SCN9AADORA2AADORA1NISCHMTOR
SCHEMBL7465829 0.67 ALDH1A1 (0.37) SCN9AKDM4EALDH1A1
SCHEMBL16369738 0.65
SCHEMBL4599509 0.64
SCHEMBL2667493 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1817030-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS Kalypsys, Inc. (US) 2007-08-15 EP disclosed
WO-2006060424-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS KALYPSYS, INC. (US) 2006-06-08 WO disclosed