SCHEMBL5200449

SCHEMBL5200449

Cc1cc(CC=O)nc(-c2ncc[nH]2)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.37
HSF1 Q00613 2/20 0.35
NISCH Q9Y2I1 2/20 0.35
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 2/20 0.33
FFAR1 O14842 1/20 0.32
ADORA2A P29274 1/20 0.31
ADORA1 P30542 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
SMPD3 Q9NY59 1/20 0.31
PDE4A P27815 1/20 0.30
PDE4B Q07343 1/20 0.30
PDE4C Q08493 1/20 0.30
PDE4D Q08499 1/20 0.30
MTOR P42345 1/20 0.30
ADK P55263 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5199466 0.72 LMNA (0.46) BRD4HSF1NISCHALDH1A1KDM4E
SCHEMBL5201542 0.70 FFAR1 (0.39) NISCHHCRTR1HCRTR2ALDH1A1FFAR1
SCHEMBL30307673 0.69 SLC6A3 (0.41) ALDH1A1
SCHEMBL5201190 0.68 MAPK14 (0.33) HCRTR1HCRTR2ALDH1A1KDM4E
SCHEMBL9026316 0.68 NISCH (0.50) BRD4HSF1NISCHALDH1A1KDM4E
SCHEMBL5201877 0.68 NUDT1 (0.35) BRD4NISCHALDH1A1KDM4EADORA2A
SCHEMBL5200348 0.68 NISCH (0.34) BRD4HSF1NISCHHCRTR1HCRTR2
SCHEMBL5200333 0.67 KDM4E (0.39) BRD4HSF1NISCHHCRTR1HCRTR2
SCHEMBL5204329 0.66 KDM4E (0.39) BRD4HSF1NISCHHCRTR1HCRTR2
SCHEMBL875422 0.66 NOS2 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1817030-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS Kalypsys, Inc. (US) 2007-08-15 EP disclosed
WO-2006060424-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS KALYPSYS, INC. (US) 2006-06-08 WO disclosed