SCHEMBL5202219

SCHEMBL5202219

Cc1cccc(-c2ccc(-n3cnc(C(N)=O)c3N)cc2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RIPK2 O43353 2/20 0.44
DHODH Q02127 3/20 0.41
TLR8 Q9NR97 2/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
CSF1R P07333 1/20 0.39
FLT1 P17948 1/20 0.39
FLT3 P36888 1/20 0.39
MAP4K4 O95819 1/20 0.39
XDH P47989 1/20 0.38
PARP1 P09874 1/20 0.38
HSD17B1 P14061 1/20 0.38
HSD17B2 P37059 1/20 0.38
HDAC2 Q92769 1/20 0.38
GRM1 Q13255 1/20 0.38
BACE1 P56817 1/20 0.37
LIMK1 P53667 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12391453 0.82 ALDH1A1 (0.49) ALDH1A1LMNAXDHGRM1NPC1
SCHEMBL5447368 0.80 KDR (0.52) CSF1RFLT1FLT3MAP4K4LIMK1
SCHEMBL4877916 0.72 ALDH1A1 (0.41) ALDH1A1LMNANPC1RAB9AKMT2A
SCHEMBL5447338 0.70 KDR (0.55) CSF1RFLT1FLT3MAP4K4NPC1
SCHEMBL12394209 0.70 DHODH (0.64) DHODHCSF1RFLT1FLT3PARP1
SCHEMBL6508388 0.69 ITK (0.47) ALDH1A1LMNACSF1RFLT1FLT3
SCHEMBL5201463 0.69 KDR (0.41) ALDH1A1LMNACSF1RFLT1FLT3
SCHEMBL19878461 0.69 MKNK1 (0.47) RIPK2DHODHTLR8CSF1RFLT3
SCHEMBL5440835 0.69 KDR (0.53) LMNACSF1RFLT1FLT3NPC1
SCHEMBL3534998 0.68 ALDH1A1 (0.46) ALDH1A1LMNAKMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761503-A2 IMIDAZOL DERIVATIVES AS TYROSINE KINASE INHIBITORS MERCK PATENT GmbH (DE) 2007-03-14 EP disclosed
WO-2005097755-A2 IMIDAZOL DERIVATIVES AS TYROSINE KINASE INHIBITORS MERCK PATENT GMBH (DE) 2005-10-20 WO disclosed