SCHEMBL5202464

SCHEMBL5202464

CC(C)(C)OC(=O)NCc1cccc(Oc2ccccc2N(Cc2ccc(-c3ccccc3)cc2)C(=O)CCCC(=O)NCc2ccccc2F)c1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
POLB P06746 2/20 0.41
LMNA P02545 1/20 0.41
HTT P42858 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
KDM4E B2RXH2 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.39
HDAC1 Q13547 1/20 0.37
SRC P12931 1/20 0.35
NR3C1 P04150 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ACHE P22303 1/20 0.35
HPGD P15428 1/20 0.35
TSPO P30536 1/20 0.35
CYP3A4 P08684 1/20 0.35
GLS O94925 1/20 0.35
PTPN1 P18031 1/20 0.35
EPHX2 P34913 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5204311 0.96 ALDH1A1 (0.42) ALDH1A1POLBLMNAHTTNPSR1
SCHEMBL5204997 0.94 ALDH1A1 (0.43) ALDH1A1POLBLMNAHTTNPSR1
SCHEMBL5206214 0.89 ALDH1A1 (0.40) ALDH1A1POLBLMNAHTTNPSR1
SCHEMBL5206192 0.88 HDAC1 (0.40) ALDH1A1HTTNPSR1HDAC1SMN1; SMN2
SCHEMBL5203418 0.88 ALDH1A1 (0.40) ALDH1A1POLBLMNAHTTNPSR1
Hydrochloric Acid SCHEMBL5205985 0.87 SSTR5 (0.42) ALDH1A1POLBLMNAHTTNPSR1
SCHEMBL5208000 0.86 HDAC1 (0.44) HDAC1NR3C1TSPOGLS
SCHEMBL5204960 0.82 HTT (0.37) ALDH1A1POLBLMNAHTTNPSR1
Hydrochloric Acid SCHEMBL5203571 0.82 SSTR5 (0.43) ALDH1A1POLBLMNAHTTNPSR1
SCHEMBL5204994 0.82 ALDH1A1 (0.40) ALDH1A1POLBLMNAHTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7160887-B1 Aromatic amine derivatives, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-01-09 US disclosed
EP-1123918-B1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME TAKEDA PHARMACEUTICAL (JP) 2005-03-09 EP disclosed
EP-1123918-A1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME Takeda Chemical Industries, Ltd. (JP) 2001-08-16 EP disclosed